Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 11753
TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644966BDBM644966(US20240010634, Example 21)
Affinity DataIC50: 7.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644926BDBM644926(US20240010634, Example 3)
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644967BDBM644967(US20240010634, Example 22)
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644933BDBM644933(US20240010634, Example 6)
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644977BDBM644977(US20240010634, Example 32)
Affinity DataIC50: 14.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644957BDBM644957(US20240010634, Example 12)
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644951BDBM644951(US20240010634, Example 10)
Affinity DataIC50: 15.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644964BDBM644964(US20240010634, Example 19)
Affinity DataIC50: 15.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644972BDBM644972(US20240010634, Example 27)
Affinity DataIC50: 15.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644969BDBM644969(US20240010634, Example 24)
Affinity DataIC50: 15.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644963BDBM644963(US20240010634, Example 18)
Affinity DataIC50: 16.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644970BDBM644970(US20240010634, Example 25)
Affinity DataIC50: 16.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644934BDBM644934(US20240010634, Example 7)
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644971BDBM644971(US20240010634, Example 26)
Affinity DataIC50: 17.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644974BDBM644974(US20240010634, Example 29)
Affinity DataIC50: 17.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644968BDBM644968(US20240010634, Example 23)
Affinity DataIC50: 18.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644960BDBM644960(US20240010634, Example 15)
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644943BDBM644943(US20240010634, Example 8)
Affinity DataIC50: 19.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644965BDBM644965(US20240010634, Example 20)
Affinity DataIC50: 21.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644925BDBM644925(US20240010634, Example 4 | US20240010634, Example ...)
Affinity DataIC50: 21.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644930BDBM644930(US20240010634, Example 5)
Affinity DataIC50: 26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644978BDBM644978(US20240010634, Example 33)
Affinity DataIC50: 26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644956BDBM644956(US20240010634, Example 11)
Affinity DataIC50: 26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644950BDBM644950(US20240010634, Example 9)
Affinity DataIC50: 26.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644973BDBM644973(US20240010634, Example 28)
Affinity DataIC50: 26.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644958BDBM644958(US20240010634, Example 13)
Affinity DataIC50: 30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644976BDBM644976(US20240010634, Example 31)
Affinity DataIC50: 30.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644924BDBM644924(US20240010634, Example 1)
Affinity DataIC50: 33.2nMAssay Description:IC50s were determined using the in vitro HotSpot kinase assay (purified enzymes, 33P-ATP, an appropriate substrate and 1 μM ATP.).More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644925BDBM644925(US20240010634, Example 4 | US20240010634, Example ...)
Affinity DataIC50: 34.5nMAssay Description:IC50s were determined using the in vitro HotSpot kinase assay (purified enzymes, 33P-ATP, an appropriate substrate and 1 μM ATP.).More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644962BDBM644962(US20240010634, Example 17)
Affinity DataIC50: 37.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644959BDBM644959(US20240010634, Example 14)
Affinity DataIC50: 64nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644975BDBM644975(US20240010634, Example 30)
Affinity DataIC50: 75.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent

TargetActivated CDC42 kinase 1(Human)
H. Lee Moffitt Cancer Center and Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 644961BDBM644961(US20240010634, Example 16)
Affinity DataIC50: 149nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2024
Entry Details
US Patent