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Report error Found 230 Enz. Inhib. hit(s) with all data for entry = 11773
LigandPNGBDBM645890(US20240018157, Example 92)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645895(US20240018157, Example 97)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645902(Step 1: N-(5-(difluoromethyl)-6-(2H-1,2,3-triazol-...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645914(Step 1: 2-(difluoromethyl)-1-fluoro-4-nitrobenzene...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645920((R)-2-chloro-N-(5-(difluoromethyl)-6-(dimethylcarb...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645923((R)-2-fluoro-8-methyl-N-(5-methyl-6-(2H-1,2,3-tria...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645924(Step 1: Mixture of methyl 2-(5-bromo-3-(difluorome...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645925(US20240018157, Example 127)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645926(Step 1: 1-(tert-butyl) 3-ethyl 3-methyl-4-oxopyrro...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645934(Step 1: tert-butyl 2-chloro-3-fluoro-8-methyl-8-(t...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645938(US20240018157, Example 140)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645944(Step 1: tert-butyl 3-fluoro-8-methyl-8-(trifluorom...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645947((R)-2-chloro-N-(5-(difluoromethyl)-6-(ethyl(methyl...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645948((R)-2-chloro-N-(6-(cyclopropylcarbamoyl)-5-(difluo...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645949(US20240018157, Example 151)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645950(Step 1: 3-chloro-5-isocyanato-2-(2H-1,2,3-triazol-...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645979((R)—N-(6-(2H-1,2,3-triazol-2-yl)-5-(trifluoro...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645989((8R)—N-(5-(difluoromethyl)-6-(4-(1-hydroxyeth...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645999(US20240018157, Example 201)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM646003(US20240018157, Example 205)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645800(2-chloro-N-(5-chloro-6-(2H-1,2,3-triazol-2-yl)pyri...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645802(US20240018157, Example 4)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645803(Step 1: 1-(tert-butyl) 4-ethyl 4-methyl-3-oxopiper...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645805(2-chloro-N-(5-chloro-6-(2H-1,2,3-triazol-2-yl)pyri...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645808(N-(5-chloro-6-(2H-1,2,3-triazol-2-yl)pyridin-3-yl)...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645810(US20240018157, Example 12)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645814(US20240018157, Example 16)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645814(US20240018157, Example 16)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645816((R)-2-chloro-N-(5-chloro-6-methoxypyridin-3-yl)-8-...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645816((R)-2-chloro-N-(5-chloro-6-methoxypyridin-3-yl)-8-...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645817(US20240018157, Example 19)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645819((R)-2-chloro-8-methyl-N-(5-methyl-6-(2H-1,2,3-tria...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM645819((R)-2-chloro-8-methyl-N-(5-methyl-6-(2H-1,2,3-tria...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645822((R)-2-chloro-N-(5-chloro-6-(4-(hydroxymethyl)-2H-1...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645822((R)-2-chloro-N-(5-chloro-6-(4-(hydroxymethyl)-2H-1...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645823(US20240018157, Example 25)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645823(US20240018157, Example 25)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645824(US20240018157, Example 26)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645824(US20240018157, Example 26)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645825(US20240018157, Example 27)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645825(US20240018157, Example 27)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645827((R)-2-chloro-N-(5-chloro-6-(4-((dimethylamino)meth...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645830(US20240018157, Example 32)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645830(US20240018157, Example 32)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645832(US20240018157, Example 34)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645833((R)-2-chloro-N-(5-(difluoromethyl)-6-(2H-1,2,3-tri...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM645833((R)-2-chloro-N-(5-(difluoromethyl)-6-(2H-1,2,3-tri...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645834((R)-2-chloro-N-(5-(difluoromethyl)-6-(1H-1,2,3-tri...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645834((R)-2-chloro-N-(5-(difluoromethyl)-6-(1H-1,2,3-tri...)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 1 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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LigandPNGBDBM645837(US20240018157, Example 39)
Affinity DataIC50: <10nMAssay Description:The final assay buffer includes 2 nM of MALT1 full-length protein, 50 μM Ac-LRSR-AMC substrate, 50 mM Tris pH 7.5, 600 mM Sodium Citrate, 1 mM D...More data for this Ligand-Target Pair
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