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Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 11924
TargetBromodomain-containing protein 4 [368-440](Human)
Chia Tai Tianqing Pharmaceutical Group Co.

US Patent
LigandPNGBDBM661115(US20240101551, Compound of Formula I)
Affinity DataIC50:  0.25nMAssay Description:In the present application, the IC50 value of the compound of formula (I) in inhibiting BRD4 (BD1) enzyme binding reaction were determined by homogen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetBromodomain-containing protein 4 [75-147](Human)
Chia Tai Tianqing Pharmaceutical Group Co.

US Patent
LigandPNGBDBM661115(US20240101551, Compound of Formula I)
Affinity DataIC50:  0.640nMAssay Description:In the present application, the IC50 value of the compound of formula (I) in inhibiting BRD4 (BD1) enzyme binding reaction were determined by homogen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent