Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 11930
LigandPNGBDBM661913(US20240101589, Example 11)
Affinity DataIC50: 6nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661908((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 6nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661932((1R,2S,3R,5R)-3- {4-amino-5-chloro- 7H-pyrrolo[2,3...)
Affinity DataIC50: 6.10nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661931((1R,2S,3R,5R)-3- {4-amino-5-fluoro- 7H-pyrrolo[2,3...)
Affinity DataIC50: 6.10nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661933((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 6.10nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661922(US20240101589, Example 20)
Affinity DataIC50: 6.10nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661934((1R,2S,3R,5R)-3- {4-amino-7H- pyrrolo[2,3- d]pyrim...)
Affinity DataIC50: 6.22nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661935((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 8.24nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661936((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 9.11nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661929(US20240101589, Example 27)
Affinity DataIC50: 9.60nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661924(US20240101589, Example 22)
Affinity DataIC50: 12.8nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661930(US20240101589, Example 28)
Affinity DataIC50: 19.7nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661906((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 22.7nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661923(US20240101589, Example 21)
Affinity DataIC50: 23.9nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661904((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 42.6nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661903(US20240101589, Example 1 | US20240101589, Example ...)
Affinity DataIC50: 44.8nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661914(US20240101589, Example 12)
Affinity DataIC50: 46.6nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661943(US20240101589, Example 41)
Affinity DataIC50: 60nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661927(US20240101589, Example 23)
Affinity DataIC50: 63.5nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661937((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 63.7nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661938((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 103nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661939((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 117nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661911(US20240101589, Example 9)
Affinity DataIC50: 123nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661912(US20240101589, Example 10)
Affinity DataIC50: 150nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661903(US20240101589, Example 1 | US20240101589, Example ...)
Affinity DataIC50: 196nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661926((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 231nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661905((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 317nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661917((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 351nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661928((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 351nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661916((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 413nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661918((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 453nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661915((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 460nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661910((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 505nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661921((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 522nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661909((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 568nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661925((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 1.09E+3nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661919((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 1.31E+3nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661940(3-{4-amino-5-bromo- 7H-pyrrolo[2,3- d]pyrimidin-7-...)
Affinity DataIC50: 2.64E+3nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661920((2R,3R,4S,5R)-2- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 2.93E+3nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661941((1R,2S,3R,5R)-3- {4-amino-5-bromo- 7H-pyrrolo[2,3-...)
Affinity DataIC50: 3.01E+3nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent

LigandPNGBDBM661942(3-[(1R,2R,3S,4R)- 4-{4-amino-5- bromo-7H-pyrrolo[2...)
Affinity DataIC50: 7.93E+3nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2024
Entry Details
US Patent