Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 12010
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669889((S, 13E, 14E)-2-ethyl-45-fluoro-6-methyl-9-oxo-5,8...)
Affinity DataIC50:  0.420nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669889((S, 13E, 14E)-2-ethyl-45-fluoro-6-methyl-9-oxo-5,8...)
Affinity DataIC50:  0.930nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669890((S, 13E, 14E)-12-amino-2-ethyl-45-fluoro-6-methyl-...)
Affinity DataIC50:  1.80nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669888( Example 5 of WO2019023417A1 | US20240132517, Exam...)
Affinity DataIC50:  1.80nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
PDB3D3D Structure (crystal)

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669890((S, 13E, 14E)-12-amino-2-ethyl-45-fluoro-6-methyl-...)
Affinity DataIC50:  2.20nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669888( Example 5 of WO2019023417A1 | US20240132517, Exam...)
Affinity DataIC50:  7.5nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
PDB3D3D Structure (crystal)

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669888( Example 5 of WO2019023417A1 | US20240132517, Exam...)
Affinity DataIC50:  10nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent


TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669889((S, 13E, 14E)-2-ethyl-45-fluoro-6-methyl-9-oxo-5,8...)
Affinity DataIC50:  15nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669890((S, 13E, 14E)-12-amino-2-ethyl-45-fluoro-6-methyl-...)
Affinity DataIC50:  30nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669891(US20240132517, Comparative Compound 42)
Affinity DataIC50:  85nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669891(US20240132517, Comparative Compound 42)
Affinity DataIC50:  289nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669891(US20240132517, Comparative Compound 42)
Affinity DataIC50: >1.00E+4nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent