Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 12060 Sort by
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675070(US20240158406, Compound 3-I)
Affinity DataIC50: 10nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675072((S)-4-(trifluoromethyl)-5-((1-((5-(5-(trifluoromet...)
Affinity DataIC50: 10nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675075((S)-5-((1-((3-chloro-5-(5-(trifluoromethyl)pyrazin...)
Affinity DataIC50: 10nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675076(US20240158406, Compound 21)
Affinity DataIC50: 10nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM431646(5-[[(2S)-1-(3-Oxo-3-[4-[5-(trifluoromethyl)pyrimid...)
Affinity DataIC50: 20nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675069((S)-4-(trifluoromethyl)-5-((1-((5-(5-(5-(trifluoro...)
Affinity DataIC50: 30nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675073((S)-4-(trifluoromethyl)-5-((1-((7-(5-(trifluoromet...)
Affinity DataIC50: 30nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675074((S)-5-((1-((3-chloro-5-(5-(trifluoromethyl)pyrimid...)
Affinity DataIC50: 30nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675071(US20240158406, Compound 3-II)
Affinity DataIC50: 75nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675069((S)-4-(trifluoromethyl)-5-((1-((5-(5-(5-(trifluoro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM431646(5-[[(2S)-1-(3-Oxo-3-[4-[5-(trifluoromethyl)pyrimid...)
Affinity DataIC50: 3.90E+3nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM431646(5-[[(2S)-1-(3-Oxo-3-[4-[5-(trifluoromethyl)pyrimid...)
Affinity DataIC50: 1.00E+4nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675069((S)-4-(trifluoromethyl)-5-((1-((5-(5-(5-(trifluoro...)
Affinity DataIC50: 1.00E+4nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675069((S)-4-(trifluoromethyl)-5-((1-((5-(5-(5-(trifluoro...)
Affinity DataIC50: 1.00E+4nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM431646(5-[[(2S)-1-(3-Oxo-3-[4-[5-(trifluoromethyl)pyrimid...)
Affinity DataIC50: 1.00E+4nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
Chengdu Baiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM675069((S)-4-(trifluoromethyl)-5-((1-((5-(5-(5-(trifluoro...)
Affinity DataIC50: 1.00E+4nMAssay Description:This assay adopted PARP1, TNKS1, TNKS2, PARP7 and PARP14 chemiluminescence detection kits (BPS, Cat No. 80551/80552/80573/80578/79729/80568) for enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent