Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 12067
TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674311BDBM674311(US20240165139, Compound 43)
Affinity DataIC50: 106nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674312BDBM674312(US20240165139, Compound 44)
Affinity DataIC50: 136nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674298BDBM674298(US20240165139, Compound 17)
Affinity DataIC50: 150nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674299BDBM674299(US20240165139, Compound 18)
Affinity DataIC50: 170nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674300BDBM674300(US20240165139, Compound 24)
Affinity DataIC50: 190nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674313BDBM674313(US20240165139, Compound 46)
Affinity DataIC50: 192nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 528659BDBM528659(US11197877, Compound 20 | US20240165139, Compound ...)
Affinity DataIC50: 240nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674308BDBM674308(US20240165139, Compound 34)
Affinity DataIC50: 340nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674309BDBM674309(US20240165139, Compound 36)
Affinity DataIC50: 510nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 528660BDBM528660(US11197877, Compound 21 | US20240165139, Compound ...)
Affinity DataIC50: 520nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674302BDBM674302(US20240165139, Compound 19)
Affinity DataIC50: 580nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674301BDBM674301(US20240165139, Compound 25)
Affinity DataIC50: 660nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674310BDBM674310(US20240165139, Compound 35)
Affinity DataIC50: 720nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 528663BDBM528663(US11197877, Compound 33 | US20240165139, Compound ...)
Affinity DataIC50: 2.12E+3nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674306BDBM674306(US20240165139, Compound 31)
Affinity DataIC50: 2.36E+3nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent

TargetE-selectin(Human)
Glycomimetics

US Patent
LigandChemical structure of BindingDB Monomer ID 674305BDBM674305(US20240165139, Compound 30)
Affinity DataIC50: 2.78E+3nMAssay Description:The inhibition assay to screen for and characterize glycomimetic antagonists of E-selectin is a competitive binding assay, which allows the determina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2024
Entry Details
US Patent