Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 12164
TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683342BDBM683342(US20240217973, Compound 001)
Affinity DataIC50: 0.710nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683353BDBM683353(US20240217973, Compound 011)
Affinity DataIC50: 1.57nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683343BDBM683343(US20240217973, Compound 002)
Affinity DataIC50: 1.65nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683345BDBM683345(US20240217973, Compound 003B)
Affinity DataIC50: 1.90nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683346BDBM683346(US20240217973, Compound 004)
Affinity DataIC50: 2.46nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683351BDBM683351(US20240217973, Compound 009)
Affinity DataIC50: 2.80nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683347BDBM683347(US20240217973, Compound 005)
Affinity DataIC50: 2.85nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683352BDBM683352(US20240217973, Compound 010)
Affinity DataIC50: 3.04nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683344BDBM683344(US20240217973, Compound 003A)
Affinity DataIC50: 4.40nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683348BDBM683348(US20240217973, Compound 006)
Affinity DataIC50: 13.6nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683349BDBM683349(US20240217973, Compound 007)
Affinity DataIC50: 16nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 683350BDBM683350(US20240217973, Compound 008)
Affinity DataIC50: 36.5nMAssay Description:1× buffer preparation (which was prepared and used immediately): Kinase assay buffer III was diluted with ddH2O to 1× assay buffer for later use.The ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
US Patent