Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 12353
TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi)

US Patent
LigandPNGBDBM697147(US20240309018, Compound WX001)
Affinity DataIC50: 0.540nMAssay Description:1. Purpose of the Assay:The ability of the compound to inhibit ERK1 and ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/16/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 3(Human)
D3 Bio (Wuxi)

US Patent
LigandPNGBDBM697147(US20240309018, Compound WX001)
Affinity DataIC50: 1.40nMAssay Description:1. Purpose of the Assay:The ability of the compound to inhibit ERK1 and ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/16/2025
Entry Details
US Patent