Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 12472
TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704703(3-Hydroxy-5- (3-m-tolylisoxazol-5- yl)picolinoyl g...)
Affinity DataIC50: 133nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704707(3-Hydroxy-5-(3-m- bromophenylisoxazol- 5-yl)picoli...)
Affinity DataIC50: 233nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704706(3-Hydroxy-5-(3-m- chlorophenylisoxazol- 5-yl)picol...)
Affinity DataIC50: 247nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704720(3-Hydroxy-5-(3-m- dichlorophenylisoxazol- 5-yl)pic...)
Affinity DataIC50: 285nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704716(3-Hydroxy-5-(3-m- dimethylphenylisoxazol- 5-yl)pic...)
Affinity DataIC50: 324nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704711(3-Hydroxy-5-(3-m- trifluoromethylphenylisoxazol-5-...)
Affinity DataIC50: 336nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704702(3-Hydroxy-5- (3-phenylisoxazol-5- yl)picolinoyl gl...)
Affinity DataIC50: 369nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704719(3-Hydroxy-5-(3- p-chlorophenylisoxazol- 5-yl)picol...)
Affinity DataIC50: 393nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704715(3-Hydroxy-5- (3-p-tolylisoxazol- 5-yl)picolinoyl g...)
Affinity DataIC50: 424nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704705(3-Hydroxy-5-(3-m- methoxyphenylisoxazol- 5-yl)pico...)
Affinity DataIC50: 432nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704718(3-Hydroxy-5-(3- o-chlorophenylisoxazol- 5-yl)picol...)
Affinity DataIC50: 436nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704722(3-Hydroxy-5-(3- p-bromophenylisoxazol- 5-yl)picoli...)
Affinity DataIC50: 436nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704714(3-Hydroxy-5- (3-o-tolylisoxazol- 5-yl)picolinoyl g...)
Affinity DataIC50: 449nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704712(3-Hydroxy-5-(3- (naphthyl-1-yl)isoxazol- 5-yl)pico...)
Affinity DataIC50: 488nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704727(3-Hydroxy-5-(3-m- difluorophenylisoxazol- 5-yl)pic...)
Affinity DataIC50: 489nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704717(3-Hydroxy-5-(3- m-fluorophenylisoxazol- 5-yl)picol...)
Affinity DataIC50: 533nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704726(3-Hydroxy-5-(3- p-fluorophenylisoxazol- 5-yl)picol...)
Affinity DataIC50: 540nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704724(3-Hydroxy-5-(3-p- trifluoromethylphenylisoxazol- 5...)
Affinity DataIC50: 555nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704708(3-Hydroxy-5-(3- cyclohexylisoxazol-5- yl)picolinoy...)
Affinity DataIC50: 648nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704721(3-Hydroxy-5-(3- o-bromophenylisoxazol- 5-yl)picoli...)
Affinity DataIC50: 691nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704728(3-Hydroxy-5-(3-m-tert- butylphenylisoxazol 5-yl)pi...)
Affinity DataIC50: 782nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704734(3-Hydroxy-5- (3,4-diphenylisoxazol- 5-yl)picolinoy...)
Affinity DataIC50: 787nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704725(3-Hydroxy-5-(3-o- fluorophenylisoxazol- 5-yl)picol...)
Affinity DataIC50: 799nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704709(3-Hydroxy-5-(3- cyclopropylisoxazol-5- yl)picolino...)
Affinity DataIC50: 907nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704710(3-Hydroxy-5-(3-m- cyanophenylisoxazol- 5-yl)picoli...)
Affinity DataIC50: 944nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704729(3-Hydroxy-5-(3- phenylisoxazol-5-yl)-6- methylpico...)
Affinity DataIC50: 991nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704733(3-Hydroxy-5- (4-cyclohexyl-3- phenylisoxazol-5-yl)...)
Affinity DataIC50: 998nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704730(3-Hydroxy-5-(4- methyl-3-phenylisoxazol- 5-yl)pico...)
Affinity DataIC50: 1.01E+3nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704731(3-Hydroxy-5-(4-tert-butyl-3- phenylisoxazol- 5-yl)...)
Affinity DataIC50: 1.21E+3nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704723(3-Hydroxy-5-(3-o- trifluoromethylphenylisoxazol- 5...)
Affinity DataIC50: 1.35E+3nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704704(3-Hydroxy-5- (3-biphenylisoxazol-5- yl)picolinoyl ...)
Affinity DataIC50: 1.80E+3nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704713(3-Hydroxy-5-(3- (naphthyl-2-yl)isoxazol- 5-yl)pico...)
Affinity DataIC50: 1.83E+3nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM704732(3-Hydroxy-5-(4-cyclopropyl-3- phenylisoxazol- 5-yl...)
Affinity DataIC50: 1.92E+3nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

TargetEgl nine homolog 1/Hypoxia-inducible factor 1-alpha [788-822](Human)
China Pharmaceutical University

US Patent
LigandPNGBDBM107704(US8598210, Table XV, 11 | US8598210, 119 | US87228...)
Affinity DataIC50: 2.90E+4nMAssay Description:The ability of the compounds to compete with a fluorophore-labeled HIF-la peptide fragment (FITC-HIF-1α 788-822) for binding to the PHD2 protein was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent