Compile Data Set for Download or QSAR
Report error Found 253 Enz. Inhib. hit(s) with all data for entry = 12498
LigandPNGBDBM706860((R)-7-(1-(6- (trifluoromethyl)pyridin-3- yl)piperi...)
Affinity DataKi:  2.80nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706895(6-((1r,4r)-4-(3,4- difluorophenyl)cyclohexyl)-2- t...)
Affinity DataKi:  6.5nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706896(6-((1s,4s)-4-(3,4- difluorophenyl)cyclohexyl)-2- t...)
Affinity DataKi:  6.70nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706780(6-((1R,3S)-3-(1-isopropyl-3-(5- (trifluoromethyl)p...)
Affinity DataKi:  6.90nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706886(6-((1s,4s)-4-(2-isopropyl-6- (trifluoromethyl)pyri...)
Affinity DataKi:  8nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706903(7-((1s,4s)-4-(3,4- difluorophenyl)cyclohexyl)-2- t...)
Affinity DataKi:  8nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706839(6-(1-(3-cyclopropyl-5- (trifluoromethyl)pyridin-2-...)
Affinity DataKi:  9nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706848(6-((1s,4s)-4-(3-chloro-5- (trifluoromethyl)pyridin...)
Affinity DataKi:  9.60nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706853(6-((1R,3S)-3-(1-isopropyl-3-(4- (trifluoromethyl)p...)
Affinity DataKi:  9.90nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706765(6-(1-(3-methyl-5- (trifluoromethyl)pyridin-2- yl)p...)
Affinity DataKi:  10nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706854(6-((1S,3R)-3-(1-isopropyl-3-(4- (trifluoromethyl)p...)
Affinity DataKi:  10nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706756(6-((1R,3S)-3-(4- (trifluoromethyl)phenyl)cyclopen-...)
Affinity DataKi:  11nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706810(6-((1r,4r)-4-(1-cyclobutyl-5- (trifluoromethyl)-1H...)
Affinity DataKi:  11nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706821(6-(1-(3-fluoro-5- (trifluoromethyl)pyridin-2- yl)p...)
Affinity DataKi:  11nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706845(6-((1s,4s)-4-(3-methyl-5- (trifluoromethyl)pyridin...)
Affinity DataKi:  11nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706845(6-((1s,4s)-4-(3-methyl-5- (trifluoromethyl)pyridin...)
Affinity DataKi:  11nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706901(6-((1r,4r)-4-(2-cyclopropyl-6- (trifluoromethyl)py...)
Affinity DataKi:  11nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706809(6-((1r,4r)-4-(1-cyclobutyl-3- (trifluoromethyl)-1H...)
Affinity DataKi:  12nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706814((R)-7-((1r,4R)-4-(1-methyl-3- (trifluoromethyl)-1H...)
Affinity DataKi:  12nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706844(7-((1S,3S)-3-(1-isopropyl-3-(6- (trifluoromethyl)p...)
Affinity DataKi:  12nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706852(6-((1S,3S)-3-(1-isopropyl-3-(4- (trifluoromethyl)p...)
Affinity DataKi:  12nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706884(6-((1s,4s)-4-(2-ethyl-6- (trifluoromethyl)pyridin-...)
Affinity DataKi:  12nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706922(6-((1r,4r)-4-(5-chloro-2- (trifluoromethyl)pyridin...)
Affinity DataKi:  12nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706819(6-(1-(3-chloro-5- (trifluoromethyl)pyridin-2- yl)p...)
Affinity DataKi:  13nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706843(7-((1R,3S)-3-(1-isopropyl-3-(6- (trifluoromethyl)p...)
Affinity DataKi:  13nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706806((R)-6-(1-(4- (trifluoromethyl)phenyl)piperi- din-3...)
Affinity DataKi:  14nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706850(6-((1s,4s)-4-(2-methyl-6- (trifluoromethyl)pyridin...)
Affinity DataKi:  14nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706861((S)-7-(1-(6- (trifluoromethyl)pyridin-3- yl)piperi...)
Affinity DataKi:  14nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706885(6-((1r,4r)-4-(2-isopropyl-6- (trifluoromethyl)pyri...)
Affinity DataKi:  14nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706754(6-((1S,3R)-3-(4- (trifluoromethyl)phenyl)cyclopen-...)
Affinity DataKi:  14.8nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706757(6-((1S,3S)-3-(4- (trifluoromethyl)phenyl)cyclopen-...)
Affinity DataKi:  15nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706780(6-((1R,3S)-3-(1-isopropyl-3-(5- (trifluoromethyl)p...)
Affinity DataKi:  15nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706781(6-((1S,3R)-3-(1-isopropyl-3-(5- (trifluoromethyl)p...)
Affinity DataKi:  15nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706883(6-((1r,4r)-4-(2-ethyl-6- (trifluoromethyl)pyridin-...)
Affinity DataKi:  15nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706920(7-((1r,4r)-4-(1-(tert-butyl)-3- (trifluoromethyl)-...)
Affinity DataKi:  15nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706760(6-((1r,4r)-4-(4- (trifluoromethyl)phenyl)cyclo hex...)
Affinity DataKi:  15.8nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706766(6-((1r,4r)-4-(1-isopropyl-3- (trifluoromethyl)-1H-...)
Affinity DataKi:  16nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706846(6-((1r,4r)-4-(3-methyl-5- (trifluoromethyl)pyridin...)
Affinity DataKi:  16nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706840(6-(1-(5-fluoro-3- (trifluoromethyl)pyridin-2- yl)p...)
Affinity DataKi:  17nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706765(6-(1-(3-methyl-5- (trifluoromethyl)pyridin-2- yl)p...)
Affinity DataKi:  17.5nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706790(6-((1R,3R)-3-(1-isopropyl-3-(6- (trifluoromethyl)p...)
Affinity DataKi:  18nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706798(6-((3R,5R)-5-(4- (trifluoromethyl)phenyl)tetrahy- ...)
Affinity DataKi:  18nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706851(7-(1-(3-fluoro-5- (trifluoromethyl)pyridin-2- yl)p...)
Affinity DataKi:  18nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706770(6-((1S,3S)-3-(1-isopropyl-3- (trifluoromethyl)-1H-...)
Affinity DataKi:  18.7nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706771(6-((1R,3S)-3-(1-isopropyl-3- (trifluoromethyl)-1H-...)
Affinity DataKi:  19nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

LigandPNGBDBM706783(6-((1S,3S)-3-(1-isopropyl-3-(5- (trifluoromethyl)p...)
Affinity DataKi:  19nMAssay Description:SPA: Determination of equilibrium dissociation constant Kd of radioligand: Membrane prepared as described above was pre-incubated with PVT-WGA SPA be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706758(6-((1s,4s)-4-(1-methyl-3- (trifluoromethyl)-1H-pyr...)
Affinity DataKi:  20nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706759(6-((1r,4r)-4-(1-methyl-3- (trifluoromethyl)-1H-pyr...)
Affinity DataKi:  20nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706760(6-((1r,4r)-4-(4- (trifluoromethyl)phenyl)cyclo hex...)
Affinity DataKi:  20nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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LigandPNGBDBM706791(6-((1R,3S)-3-(1-isopropyl-3-(6- (trifluoromethyl)p...)
Affinity DataKi:  20nMAssay Description:DHCR7: The radioligand binding assay was prepared by adding assay buffer diluted hEBP-DHCR7 membrane at 66.7 μg/ml×150 μl/well into the 96-well compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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