Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 12652
TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 605701BDBM605701(US11673894, Ex. No. 79 | US20250041310, Compound 2...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533359BDBM533359(US11220510, Example 4 | US20250041310, Compound 19)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533400BDBM533400(US11220510, Example 30 | US20250041310, Compound 2...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 605662BDBM605662(US11673894, Ex. No. 41 | US20250041310, Compound 1)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 605698BDBM605698(US11673894, Ex. No. 77 | US11673894, Ex. No. 76 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522564BDBM522564(US11161850, Example 29 | US11161850, Example 127 |...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522676BDBM522676(US11161850, Example 49 | US11161850, Example 50 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 524539BDBM524539(US11168089, Ex. No. 15 | US11873304, Example 15 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 524540BDBM524540(US11168089, Ex. No. 16 | US11873304, Example 16 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 524525BDBM524525(US11168089, Ex. No. 1 | US11873304, Example 1 | US...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 524538BDBM524538(US11168089, Ex. No. 14 | US11873304, Example 14 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 605700BDBM605700(US11673894, Ex. No. 78 | US20250041310, Compound 3)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 605716BDBM605716(US11673894, Ex. No. 94 | US20250041310, Compound 4)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533344BDBM533344(US11220510, Example 2 | US20250041310, Compound 17)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533358BDBM533358(US11220510, Example 3 | US20250041310, Compound 18)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 561416BDBM561416(US11390624, Example 31 | 3-(4-amino-2-((3-fluoropy...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 561425BDBM561425(US11390624, Example 39 | 3-(4-amino-7-(1-methyl-1H...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 561401BDBM561401(US11390624, Example 16 | 3-(4-amino-2-(pyridin-2-y...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 561415BDBM561415(US11390624, Example 30 | 3-(4-amino-2-((3-fluoropy...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522719BDBM522719(US11161850, Example 77 | US20250041310, Compound 1...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522878BDBM522878(US11161850, Example 94 | US11161850, Example 95 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first seria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2025
Entry Details
US Patent