Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 12811
TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730218(US20250108123, Example II-1)
Affinity DataIC50: 0.0600nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730205(4,4'-((propane-1,3-diylbis(oxy))bis(6-methoxyisoin...)
Affinity DataIC50: 0.100nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730221(US20250108123, Example II-4)
Affinity DataIC50: 0.180nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730235(US20250108123, Example II-20)
Affinity DataIC50: 0.190nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730232(US20250108123, Example II-17)
Affinity DataIC50: 0.190nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM665306(US20240116909, Example 10 | 4-(5-(3-((2-(3-carboxy...)
Affinity DataIC50: 0.280nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730212(US20250108123, Example I-9)
Affinity DataIC50: 0.320nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730222(sodium (S)-4-(5-(3-((2-((S)-3-carboxylatobutanoyl)...)
Affinity DataIC50: 0.320nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730223(US20250108123, Example II-7)
Affinity DataIC50: 0.360nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730225(US20250108123, Example II-9)
Affinity DataIC50: 0.650nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730208(US20250108123, Example I-4)
Affinity DataIC50: 0.680nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM665304(US20240116909, Example 8 | Sodium 4-(5-(3-((2-(3-c...)
Affinity DataIC50: 1.04nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730207(US20250108123, Example I-3)
Affinity DataIC50: 1.63nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730225(US20250108123, Example II-9)
Affinity DataIC50: 2.23nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM665307(US20240116909, Example 11 | 4-(5-(3-((6-(3-carboxy...)
Affinity DataIC50: 2.54nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730209(US20250108123, Example I-5)
Affinity DataIC50: 3.28nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730233(US20250108123, Example II-18)
Affinity DataIC50: 4.59nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730220(US20250108123, Example II-3)
Affinity DataIC50: 8.40nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM665298(US20240116909, Example 2 | 4-(5-(3-((2-(3-carboxyp...)
Affinity DataIC50: 11.4nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730228(US20250108123, Example II-13)
Affinity DataIC50: 12.8nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730206(US20250108123, Example I-2)
Affinity DataIC50: 33.7nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM665309(US20240116909, Example 14 | 4-(5-(3-((2-(3-carboxy...)
Affinity DataIC50: 46.6nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730234(US20250108123, Example II-19)
Affinity DataIC50: 54.6nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730230(US20250108123, Example II-15)
Affinity DataIC50: 92.6nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730217(US20250108123, Example I-14)
Affinity DataIC50: 144nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730216(US20250108123, Example I-13)
Affinity DataIC50: 149nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM665311(US20240116909, Example 16 | 4-(5-((2-(((2-(3-carbo...)
Affinity DataIC50: 150nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730214(US20250108123, Example I-11)
Affinity DataIC50: 150nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730215(US20250108123, Example I-12)
Affinity DataIC50: 150nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730213(US20250108123, Example I-10)
Affinity DataIC50: 150nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730210(US20250108123, Example I-7)
Affinity DataIC50: 150nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730211(US20250108123, Example I-8)
Affinity DataIC50: 150nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Jacobio Pharmaceuticals Co.

US Patent
LigandPNGBDBM730236(US20250108123, Example II-21)
Affinity DataIC50: 159nMAssay Description:Cisbio Bioassays' human STING WT binding assay (#64BDSTGPEG & 64BDSTGPEH, Cisbio) is for quantitative measurement of human STING WT ligand using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent