Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 12931
TargetSortilin(Human)TBA
LigandPNGBDBM741293((2S)-5,5-dimethyl-2-[(morpholine-4-carbonyl)amino]...)
Affinity DataIC50: 260nMAssay Description:Compound affinity was determined by measuring the displacement of [3H]-neurotensin binding to h-Sortilin in SPA format. Total volume of 40 μl in 50 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetSortilin(Human)TBA
LigandPNGBDBM741294((2S)-5,5-dimethyl-2-[(1,4-oxazepane-4-carbonyl)ami...)
Affinity DataIC50: 370nMAssay Description:Compound affinity was determined by measuring the displacement of [3H]-neurotensin binding to h-Sortilin in SPA format. Total volume of 40 μl in 50 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetSortilin(Human)TBA
LigandPNGBDBM741290((2S)-2-[(benzylcarbamoyl)amino]-5,5-dimethylhexano...)
Affinity DataIC50: 380nMAssay Description:Compound affinity was determined by measuring the displacement of [3H]-neurotensin binding to h-Sortilin in SPA format. Total volume of 40 μl in 50 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetSortilin(Human)TBA
LigandPNGBDBM741291((2S)-2-{[benzyl(methyl)carbamoyl]amino}-5,5-dimeth...)
Affinity DataIC50: 430nMAssay Description:Compound affinity was determined by measuring the displacement of [3H]-neurotensin binding to h-Sortilin in SPA format. Total volume of 40 μl in 50 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetSortilin(Human)TBA
LigandPNGBDBM741292((2S)-2-{[(benzyloxy)carbonyl]amino}-5,5-dimethylhe...)
Affinity DataIC50: 560nMAssay Description:Compound affinity was determined by measuring the displacement of [3H]-neurotensin binding to h-Sortilin in SPA format. Total volume of 40 μl in 50 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent