Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 12988
LigandPNGBDBM748289(US20250186425, Example 7)
Affinity DataEC50:  55nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

LigandPNGBDBM748288(US20250186425, Example 6)
Affinity DataEC50:  550nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

LigandPNGBDBM748287(US20250186425, Example 5)
Affinity DataEC50:  550nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

LigandPNGBDBM748286(US20250186425, Example 4)
Affinity DataEC50:  550nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

LigandPNGBDBM748284(US20250186425, Example 2)
Affinity DataEC50:  550nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

LigandPNGBDBM748283(US20250186425, Example 1)
Affinity DataEC50:  550nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

LigandPNGBDBM748285(US20250186425, Example 3)
Affinity DataEC50:  5.50E+3nMAssay Description:Compound potency (EC50) and maximal extent of NCOR1 recruitment to PPARG were assessed a TR-FRET binding assay measuring association of a biotinylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent