Compile Data Set for Download or QSAR
Report error Found 158 Enz. Inhib. hit(s) with all data for entry = 13017
LigandChemical structure of BindingDB Monomer ID 50590929BDBM50590929(CHEMBL4303292 | US20240016810, Compound TABLE 16.2...)
Affinity DataIC50: 1nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50590927BDBM50590927(Apilimod | Sta-5326 | STA 5326 | STA-5326 | APILIM...)
Affinity DataIC50: 3nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645378BDBM645378(US20240016810, Compound TABLE 16.11 | US2024001681...)
Affinity DataIC50: 4.90nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645378BDBM645378(US20240016810, Compound TABLE 16.11 | US2024001681...)
Affinity DataIC50: 5nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645389BDBM645389(US20240016810, Compound TABLE 16.3 | US20240208964...)
Affinity DataIC50: 7nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50590929BDBM50590929(CHEMBL4303292 | US20240016810, Compound TABLE 16.2...)
Affinity DataIC50: 7.5nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751677BDBM751677(5-methoxy-6-(5-(1-methyl-1H-pyrazol-3-yl)pyridazin...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751676BDBM751676(5-methoxy-2-morpholino-N-(pyridin-4-yl)-6-(3-(pyri...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751699BDBM751699(2-di(pyridin-4-yl)pyrimidin-4-amine | US202501973...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751722BDBM751722(5-methoxy-6-(3-(1-methyl-1H-pyrazol-3-yl)phenyl)-N...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751674BDBM751674(5-methoxy-6-(2-(1-methyl-H-pyrazol-3-yl)pyridin-4-...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751728BDBM751728(azetidin-1-yl[4-[3-(1-methylpyrazol-3-yl)phenyl]-2...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751726BDBM751726(N,N-dimethyl-4-[3-(1-methylpyrazol-3-yl)phenyl]-2-...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751669BDBM751669(6-methoxy-6-(3-(3-methyl-1H-pyrazol-1-yl)phenyl)-2...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751668BDBM751668(6-(3-(1H-pyrazol-1-yl)phenyl)-5-methoxy-2-morpholi...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751667BDBM751667(5-methoxy-6-(5-(1-methyl-1H-pyrazol-3-yl)pyridin-3...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751673BDBM751673(6-(3,4-dimethoxyphenyl)-5-methoxy-2-morpholino-N-(...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751672BDBM751672(US20250197375, Compound 12)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751717BDBM751717(5-methoxy-2-morpholino-65-(pyridazin-3-yl)pyridin-...)
Affinity DataIC50: 10nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645377BDBM645377(US20240016810, Compound TABLE 15.2 | US20240208964...)
Affinity DataIC50: 12nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645392BDBM645392(US20240016810, Compound TABLE 16.5 | US20240208964...)
Affinity DataIC50: 14nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645401BDBM645401(US20240016810, Compound TABLE 16.14 | US2024020896...)
Affinity DataIC50: 18nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645399BDBM645399(US20240016810, Compound TABLE 16.12 | US2024020896...)
Affinity DataIC50: 18nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645402BDBM645402(US20240016810, Compound TABLE 16.15 | US2024020896...)
Affinity DataIC50: 32nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645407BDBM645407(US20240016810, Compound TABLE 16.20 | US2024020896...)
Affinity DataIC50: 42nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751701BDBM751701(6-(3-(1,4-dimethyl-1H-pyrazol-3-yl)phenyl)-6-metho...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751700BDBM751700(9-(1-methyl-1H-pyrazol-3-yl)-2-morpholino-N-(pyrid...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751700BDBM751700(9-(1-methyl-1H-pyrazol-3-yl)-2-morpholino-N-(pyrid...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751699BDBM751699(2-di(pyridin-4-yl)pyrimidin-4-amine | US202501973...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751698BDBM751698(9-(1-methyl-1H-pyrazol-3-yl)-2-morpholino-N-(pyrid...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751663BDBM751663(5-methoxy-6-(3-(1-methyl-1H-pyrazol-3-yl)phenyl)-2...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751662BDBM751662(morpholine | US20250197375, Compound 2)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751661BDBM751661(5-methoxy-2-morpholino-N-phenyl-6-(1-phenyl-1H-pyr...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751690BDBM751690(4-(5-methoxy-4-(3-(1-methyl-1H-pyrazol-3-yl)phenyl...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751734BDBM751734(6-[3-(1-methylpyrazol-3-yl)phenyl]-2-morpholino-5-...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751732BDBM751732(N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751694BDBM751694(5-methoxy-6-(3-(1-methyl-H-pyrazol-3-yl)phenyl)-N-...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751693BDBM751693(N,N-dimethyl-2-morpholino-4-(3-pyrazol-1-ylphenyl)...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751676BDBM751676(5-methoxy-2-morpholino-N-(pyridin-4-yl)-6-(3-(pyri...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751725BDBM751725(6-methyl-2-morpholino-9-pyrazol-1-yl-4-(4-pyridyla...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751675BDBM751675(4-(3-(5-methoxy-2-morpholino-6-(pyridin-4-ylamino)...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751674BDBM751674(5-methoxy-6-(2-(1-methyl-H-pyrazol-3-yl)pyridin-4-...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751728BDBM751728(azetidin-1-yl[4-[3-(1-methylpyrazol-3-yl)phenyl]-2...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751679BDBM751679(US20250197375, Compound 19)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751677BDBM751677(5-methoxy-6-(5-(1-methyl-1H-pyrazol-3-yl)pyridazin...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751667BDBM751667(5-methoxy-6-(5-(1-methyl-1H-pyrazol-3-yl)pyridin-3...)
Affinity DataIC50: 55nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751709BDBM751709(9-(1-methyl-1H-pyrazol-3-yl)-2-morpholino-N-(pyrid...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751666BDBM751666(pyrimidine-4-carboxamide | US20250197375, Compoun...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751707BDBM751707(5-methoxy-6-(3-(4-methoxy-1-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 751671BDBM751671(US20250197375, Compound 11)
Affinity DataIC50: 55nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

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