Compile Data Set for Download or QSAR
Report error Found 168 Enz. Inhib. hit(s) with all data for entry = 13053
LigandChemical structure of BindingDB Monomer ID 755087BDBM755087((R,13E,14E)-31,7-Dimethyl-17-(methylamino)-31H-5-o...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755147BDBM755147(US20250213571, Compound 99)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755090BDBM755090((7R,E)-31,7-Dimethyl-18-(methylamino)-31H-5-oxa-2,...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755089BDBM755089((R,13E,14E)-3',7-Dimethyl-17-(methylamino)-31H-5-o...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755088BDBM755088((7R,E)-3',7-Dimethyl-18-(methylamino)-31H-5-oxa-2,...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755143BDBM755143(US20250213571, Compound 95)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755142BDBM755142(US20250213571, Compound 94)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755076BDBM755076((15E,34E,7R)-32,7-dimethyl-18-(methylamino)-32H-5-...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755086BDBM755086((7R,E)-3',7-Dimethyl-18-(methylamino)-31H-5-oxa-2,...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755146BDBM755146(US20250213571, Compound 98)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755145BDBM755145(US20250213571, Compound 97)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755078BDBM755078((7R,E)-3',7-Dimethyl-18-(methylamino)-31H-5-oxa-2,...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755144BDBM755144(US20250213571, Compound 96)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755096BDBM755096(US20250213571, Compound 34)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755102BDBM755102(US20250213571, Compound 36)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755100BDBM755100(US20250213571, Compound 35)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755092BDBM755092((7R,E)-3',7-Dimethyl-18-(methylamino)-31H-5-oxa-2,...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755091BDBM755091((R,13E,14E)-3',7-Dimethyl-17-(methylamino)-31H-5-o...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755095BDBM755095(US20250213571, Compound 33)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755094BDBM755094(US20250213571, Compound 16)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755093BDBM755093(US20250213571, Compound 15)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755115BDBM755115(US20250213571, Compound 59)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755114BDBM755114(US20250213571, Compound 58)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755113BDBM755113(US20250213571, Compound 57)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755112BDBM755112(US20250213571, Compound 56)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755111BDBM755111(US20250213571, Compound 55)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755110BDBM755110(US20250213571, Compound 54)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755121BDBM755121(US20250213571, Compound 65)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755120BDBM755120(US20250213571, Compound 64)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755119BDBM755119(US20250213571, Compound 63)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755118BDBM755118(US20250213571, Compound 62)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755117BDBM755117(US20250213571, Compound 61)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755116BDBM755116(US20250213571, Compound 60)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755106BDBM755106(US20250213571, Compound 37)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755109BDBM755109(US20250213571, Compound 53)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755108BDBM755108(US20250213571, Compound 52)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755107BDBM755107(US20250213571, Compound 38)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755070BDBM755070(Synthesis of (R,13E,14E)-31,7-dimethyl-17-(methyla...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755138BDBM755138(US20250213571, Compound 90)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755068BDBM755068(Synthesis of (7R,E)-3',7-Dimethyl-18-(methylamino)...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755067BDBM755067(Synthesis of (7R,E)-7-(Hydroxymethyl)-31-methyl-18...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755141BDBM755141(US20250213571, Compound 93)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755140BDBM755140(US20250213571, Compound 92)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755073BDBM755073((7R,E)-31,7-Dimethyl-18-(methylamino)-31H-5-oxa-2,...)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755139BDBM755139(US20250213571, Compound 91)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755126BDBM755126(US20250213571, Compound 70)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755125BDBM755125(US20250213571, Compound 69)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755124BDBM755124(US20250213571, Compound 68)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755123BDBM755123(US20250213571, Compound 67)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 755122BDBM755122(US20250213571, Compound 66)
Affinity DataKd: <10nMAssay Description:Binding constants for the compounds described herein against the JH2 domain were determined by the following protocol for a KINOMEscan® assay (Discov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent

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