Compile Data Set for Download or QSAR
Report error Found 210 Enz. Inhib. hit(s) with all data for entry = 13169
TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764618BDBM764618(N-[[1-(pyrrolidin-1-ylmethyl)cyclobutyl]methyl]- |...)
Affinity DataEC50:  5.80nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764618BDBM764618(N-[[1-(pyrrolidin-1-ylmethyl)cyclobutyl]methyl]- |...)
Affinity DataEC50:  6nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764662BDBM764662(N-[[1-[(3-hydroxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  6nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764618BDBM764618(N-[[1-(pyrrolidin-1-ylmethyl)cyclobutyl]methyl]- |...)
Affinity DataEC50:  6.60nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764646BDBM764646(N-[[1-[(4-methoxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  6.60nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764638BDBM764638(N-[[1-[(4-hydroxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  7.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764662BDBM764662(N-[[1-[(3-hydroxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  7.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764652BDBM764652(N-[3-(3-methoxypiperidin-1-yl)-2,2-dimethylpropyl]...)
Affinity DataEC50:  8.10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764625BDBM764625(N-[[1-[(4-hydroxypiperidin-1-yl)methyl]cyclopentyl...)
Affinity DataEC50:  8.20nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764602BDBM764602(N-[[1-(pyrrolidin-1-ylmethyl)cyclopentyl]methyl]- ...)
Affinity DataEC50:  8.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764641BDBM764641(N-[[3-(pyrrolidin-1-ylmethyl)oxan-3-yl]methyl]-4,5...)
Affinity DataEC50:  8.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764599BDBM764599(N-[[1-[(dimethylamino)methyl]cyclopentyl]methyl]- ...)
Affinity DataEC50:  8.5nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764650BDBM764650(N-[[1-[(4-methoxy-4-methylpiperidin-1-yl)methyl]cy...)
Affinity DataEC50:  8.60nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764638BDBM764638(N-[[1-[(4-hydroxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  8.60nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764646BDBM764646(N-[[1-[(4-methoxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  8.70nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764617BDBM764617(N-[[4-(pyrrolidin-1-ylmethyl)oxan-4-yl]methyl]-4,5...)
Affinity DataEC50:  8.80nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764656BDBM764656(N-[[1-[(3-hydroxy-3-methylpiperidin-1-yl)methyl] |...)
Affinity DataEC50:  9nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764611BDBM764611(N-[[1-(azetidin-1-ylmethyl)cyclopentyl]methyl]- | ...)
Affinity DataEC50:  9.10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764629BDBM764629(N-[[3-hydroxy-1-(pyrrolidin-1-ylmethyl)cyclobutyl]...)
Affinity DataEC50:  9.10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764661BDBM764661(N-[[1-[(3-hydroxypyrrolidin-1-yl)methyl]cyclopenty...)
Affinity DataEC50:  9.10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764609BDBM764609(N-[[1-(diethylaminomethyl)cyclopentyl]methyl]-4,5,...)
Affinity DataEC50:  9.10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764633BDBM764633(N-[[1-(azetidin-1-ylmethyl)cyclobutyl]methyl]-4,5,...)
Affinity DataEC50:  9.10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764656BDBM764656(N-[[1-[(3-hydroxy-3-methylpiperidin-1-yl)methyl] |...)
Affinity DataEC50:  9.20nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764662BDBM764662(N-[[1-[(3-hydroxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  9.20nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764611BDBM764611(N-[[1-(azetidin-1-ylmethyl)cyclopentyl]methyl]- | ...)
Affinity DataEC50:  9.30nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764599BDBM764599(N-[[1-[(dimethylamino)methyl]cyclopentyl]methyl]- ...)
Affinity DataEC50:  9.30nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764625BDBM764625(N-[[1-[(4-hydroxypiperidin-1-yl)methyl]cyclopentyl...)
Affinity DataEC50:  9.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764628BDBM764628(N-[[1-[(dimethylamino)methyl]-3-hydroxycyclobutyl]...)
Affinity DataEC50:  9.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764638BDBM764638(N-[[1-[(4-hydroxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  9.40nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764620BDBM764620(N-[[1-[(dimethylamino)methyl]cyclobutyl]methyl]- |...)
Affinity DataEC50:  9.5nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764636BDBM764636(N-[[3-(pyrrolidin-1-ylmethyl)oxolan-3-yl]methyl]- ...)
Affinity DataEC50:  9.60nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764641BDBM764641(N-[[3-(pyrrolidin-1-ylmethyl)oxan-3-yl]methyl]-4,5...)
Affinity DataEC50:  9.60nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764660BDBM764660(N-[[1-[(3-hydroxypyrrolidin-1-yl)methyl]cyclopenty...)
Affinity DataEC50:  9.70nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764660BDBM764660(N-[[1-[(3-hydroxypyrrolidin-1-yl)methyl]cyclopenty...)
Affinity DataEC50:  9.80nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764635BDBM764635(N-[[3-[(dimethylamino)methyl]oxolan-3-yl]methyl]- ...)
Affinity DataEC50:  10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764625BDBM764625(N-[[1-[(4-hydroxypiperidin-1-yl)methyl]cyclopentyl...)
Affinity DataEC50:  10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764646BDBM764646(N-[[1-[(4-methoxypiperidin-1-yl)methyl]cyclobutyl]...)
Affinity DataEC50:  10nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764661BDBM764661(N-[[1-[(3-hydroxypyrrolidin-1-yl)methyl]cyclopenty...)
Affinity DataEC50:  10.2nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764602BDBM764602(N-[[1-(pyrrolidin-1-ylmethyl)cyclopentyl]methyl]- ...)
Affinity DataEC50:  10.2nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764627BDBM764627(N-[[1-[[2-hydroxyethyl(methyl)amino]methyl]cyclobu...)
Affinity DataEC50:  10.2nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764599BDBM764599(N-[[1-[(dimethylamino)methyl]cyclopentyl]methyl]- ...)
Affinity DataEC50:  10.3nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764620BDBM764620(N-[[1-[(dimethylamino)methyl]cyclobutyl]methyl]- |...)
Affinity DataEC50:  10.5nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764622BDBM764622(N-[[1-[(3-hydroxypyrrolidin-1-yl)methyl]cyclopenty...)
Affinity DataEC50:  10.5nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764624BDBM764624(N-[[1-[(3-hydroxypiperidin-1-yl)methyl]cyclopentyl...)
Affinity DataEC50:  10.8nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Mouse)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764641BDBM764641(N-[[3-(pyrrolidin-1-ylmethyl)oxan-3-yl]methyl]-4,5...)
Affinity DataEC50:  10.8nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Rat)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764636BDBM764636(N-[[3-(pyrrolidin-1-ylmethyl)oxolan-3-yl]methyl]- ...)
Affinity DataEC50:  10.9nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764643BDBM764643(N-[3-(3-hydroxypiperidin-1-yl)-2,2-dimethylpropyl]...)
Affinity DataEC50:  10.9nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764606BDBM764606(N-[2-ethyl-2-(pyrrolidin-1-ylmethyl)butyl]-4,5,6,7...)
Affinity DataEC50:  11nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764615BDBM764615(N-[[1-(pyrrolidin-1-ylmethyl)cyclohexyl]methyl]- |...)
Affinity DataEC50:  11nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetCX3C chemokine receptor 1(Human)
University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 764636BDBM764636(N-[[3-(pyrrolidin-1-ylmethyl)oxolan-3-yl]methyl]- ...)
Affinity DataEC50:  11.1nMAssay Description:Compounds (as well as stereoisomer(s) thereof and/or salt(s) thereof) were tested for CX3CR1 agonism in a cell based assay with fluorescent readout i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

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