Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 13174
TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764880(2-butyl-7-(hexahydropyridin-4-yl)-1-(3,4,5,6-tetra...)
Affinity DataEC50:  30nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764888(1-{4-[4-amino-2-butyl-1-(3,4,5,6-tetrahydro-2H-pyr...)
Affinity DataEC50:  40nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764876(2-butyl-7-methyl-1-((tetrahydro-2H-pyran-4-yl)meth...)
Affinity DataEC50:  50nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764881(2-butyl-7-(1-methylpiperidin-4-yl)-1-((tetrahydro-...)
Affinity DataEC50:  83nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764875(2-butyl-1-(piperidin-4-ylmethyl)-1H-imidazo[4,5-d]...)
Affinity DataEC50:  140nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764878(2-butyl-7-methyl-1-((1-methylpiperidin-4-yl)methyl...)
Affinity DataEC50:  200nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764865(1-(4-aminobutyl)-2-butyl-7-methyl-1H-imidazo[4,5-d...)
Affinity DataEC50:  220nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764877(2-butyl-1-[(1-methylhexahydropyridin-4-yl)methyl]t...)
Affinity DataEC50:  270nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
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TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764866(1-(4-aminobutyl)-2-butyl-1H-imidazo[4,5-d]thieno[3...)
Affinity DataEC50:  280nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764870(2-butyl-7-(1-methylpiperidin-4-yl)-1H-imidazo[4,5-...)
Affinity DataEC50:  440nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764887(2-(2-methoxyethyl)-1-[(1-methylhexahydropyridin-4-...)
Affinity DataEC50:  460nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764867(2-butyl-7-methyl-1-(piperidin-4-ylmethyl)-1H-imida...)
Affinity DataEC50:  470nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764883(2-butyl-1-((1-methylpiperidin-4-yl)methyl)-7-(tetr...)
Affinity DataEC50:  580nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764874(1-(4-((4-amino-2-butyl-7-methyl-1H-imidazo[4,5-d]t...)
Affinity DataEC50:  1.16E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764879(2-butyl-1-methyl-7-(1-methylpiperidin-4-yl)-1H-imi...)
Affinity DataEC50:  1.26E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764882(2-butyl-7-(1-methylpiperidin-4-yl)-1-((1-methylpip...)
Affinity DataEC50:  1.30E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764872(1-((1-(2-(2-(2-aminoethoxy)ethoxy)ethyl)piperidin-...)
Affinity DataEC50:  1.42E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764885(2-butyl-1-{[1-(2-methoxyethyl)hexahydropyridin-4-y...)
Affinity DataEC50:  1.43E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764886(1-(hexahydropyridin-4-ylmethyl)-2-(2-methoxyethyl)...)
Affinity DataEC50:  1.48E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764873(1-((1-(2,5,8,11,14,17,20-heptaoxadocosan-22-yl)pip...)
Affinity DataEC50:  1.69E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764868(1-(4-aminobutyl)-2-(2-methoxyethyl)-1H-imidazo[4,5...)
Affinity DataEC50:  2.41E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764871(2-butyl-7-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl...)
Affinity DataEC50:  2.50E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764869(1-(4-aminobutyl)-2-(2-ethoxymethyl)-1H-imidazo[4,5...)
Affinity DataEC50:  3.25E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 7(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764884(2-butyl-7-(hexahydropyridin-4-yl)-1-{[1-(2-methoxy...)
Affinity DataEC50:  5.05E+3nMAssay Description:1. HEK-Blue hTLR7 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 8(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764865(1-(4-aminobutyl)-2-butyl-7-methyl-1H-imidazo[4,5-d...)
Affinity DataEC50:  5.83E+3nMAssay Description:1. HEK-Blue hTLR8 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 8(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764866(1-(4-aminobutyl)-2-butyl-1H-imidazo[4,5-d]thieno[3...)
Affinity DataEC50:  8.83E+3nMAssay Description:1. HEK-Blue hTLR8 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 8(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764877(2-butyl-1-[(1-methylhexahydropyridin-4-yl)methyl]t...)
Affinity DataEC50:  1.19E+4nMAssay Description:1. HEK-Blue hTLR8 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 8(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764870(2-butyl-7-(1-methylpiperidin-4-yl)-1H-imidazo[4,5-...)
Affinity DataEC50:  1.53E+4nMAssay Description:1. HEK-Blue hTLR8 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 8(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764880(2-butyl-7-(hexahydropyridin-4-yl)-1-(3,4,5,6-tetra...)
Affinity DataEC50:  1.89E+4nMAssay Description:1. HEK-Blue hTLR8 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent

TargetToll-like receptor 8(Human)
Sichuan Kelun-Biotech Biopharmaceutical

US Patent
LigandPNGBDBM764867(2-butyl-7-methyl-1-(piperidin-4-ylmethyl)-1H-imida...)
Affinity DataEC50:  1.94E+4nMAssay Description:1. HEK-Blue hTLR8 cells (Invivogen) were cultured in DMEM medium (Hyclone) containing 10% FBS heat-inactivated fetal bovine serum (Corning). On the d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent