Compile Data Set for Download or QSAR
Report error Found 180 Enz. Inhib. hit(s) with all data for entry = 13225
TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768266BDBM768266((R)-2,3-difluoro-N-((4-((1-methylpiperidin-4-yl)ox...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768265BDBM768265((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768268BDBM768268((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768267BDBM768267((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768262BDBM768262((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768264BDBM768264(4-((R)-1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768263BDBM768263((R)-N-((4-((1-azabicyclo[2.2.1]heptan-4-yl)oxy)phe...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768258BDBM768258((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768257BDBM768257((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768260BDBM768260((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768259BDBM768259((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768254BDBM768254((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768253BDBM768253(N-((4-(((1R,4R,5R)-2-azabicyclo[2.2.1]heptan-5-yl)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768256BDBM768256((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768255BDBM768255((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768282BDBM768282((R)-2,3-difluoro-N-((1-methylpiperidin-4-yl)sulfon...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768281BDBM768281((R)-2,3-difluoro-4-(1-(5-(pyridin-2-yloxy)pyridin-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768283BDBM768283((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768278BDBM768278((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768277BDBM768277((R)-N-((4-(2-(dimethylamino)ethoxy)piperidin-1-yl)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768279BDBM768279((R)-2,3-difluoro-N-((4-methylpiperazin-1-yl)sulfon...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768273BDBM768273((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768270BDBM768270((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768269BDBM768269((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768272BDBM768272((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768271BDBM768271((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768298BDBM768298(4-((R)-1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768297BDBM768297((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768300BDBM768300((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768299BDBM768299((R)-N-((4-(2-(dimethylamino)ethoxy)phenyl)sulfonyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768294BDBM768294(4-((R)-1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768293BDBM768293((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768295BDBM768295(2,3-difluoro-N-((4-((1-methylpiperidin-3-yl)oxy)ph...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768290BDBM768290((R)-N-((4-((1-methylpiperidin-4-yl)oxy)piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768289BDBM768289((R)-N-((4-(2-(dimethylamino)ethoxy)phenyl)sulfonyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768291BDBM768291((R)-N-((4-(2-(dimethylamino)ethoxy)phenyl)sulfonyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768286BDBM768286((R)-N-((1-(dimethylamino)-2-methylpropan-2-yl)sulf...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768285BDBM768285((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768288BDBM768288((R)-N-((4-(2-(dimethylamino)ethoxy)phenyl)sulfonyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768287BDBM768287((R)-N-((4-((1-methylpiperidin-4-yl)oxy)piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768314BDBM768314((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768313BDBM768313((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768316BDBM768316((R)-N-((4-cyclohexylpiperazin-1-yl)sulfonyl)-4-(1-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768315BDBM768315((R)-N-((4-cyclopropylpiperazin-1-yl)sulfonyl)-2,3-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768310BDBM768310((R)-N-((4-ethylpiperazin-1-yl)sulfonyl)-2,3-difluo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768312BDBM768312((R)-N-((4-methylpiperazin-1-yl)sulfonyl)-4-(1-(5-(...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768311BDBM768311((R)-4-(1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768306BDBM768306(N-((4-(2-(dimethylamino)ethoxy)phenyl)sulfonyl)-2,...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768305BDBM768305(4-((R)-1-(5-(cyclopropylmethoxy)pyridin-2-yl)propo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

TargetLong-chain-fatty-acid--CoA ligase 5 [33-683](Homo sapiens (Human))
Lexicon Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 768307BDBM768307(2,3-difluoro-4-((R)-1-(5-((1R,3R)-3-methoxycyclobu...)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACSL5 enzyme activity was monitored with a coupled enzyme Amplex Red assay. The assay is carried out in 384-well microtiterplates. In a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/15/2025
Entry Details
US Patent

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