Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 13284
Targetchymase(Golden hamster)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetChymase(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetChymase(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 20nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

Targetchymase(Golden hamster)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 66nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetCathepsin G(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 140nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetCathepsin G(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 1.30E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetPlasma kallikrein(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetPlasminogen(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetCoagulation factor X(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetSerine protease 1(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetProthrombin(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetCoagulation factor XI(Human)TBA
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetCoagulation factor X(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetSerine protease 1(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetProthrombin(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetCoagulation factor XI(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetPlasma kallikrein(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetPlasminogen(Human)TBA
LigandPNGBDBM256012(US9481672, 190 | US20250302837, Example fulacimsta...)
Affinity DataIC50: 1.50E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent