Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 13290
LigandPNGBDBM637667((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637665((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637662(R-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637613((R)-(3-aminopiperidin-1-yl)(2-(1-(pyridine-2-ylmet...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637610((R)-(3-aminopiperidin-1-yl)(2-(1-(pyridin-4-ylmeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM773964((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637607((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637617((R)-(3-aminopiperidin-1-yl)(2-(1-(2-fluorobenzyl)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637614((R)-(3-aminopiperidin-1-yl)(2-(3-ethylbenzo[b]thio...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637641((R)-(3-aminopiperidin-1-yl)(2-(1-(4-methoxybenzyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM773977((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637659(R-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637657((R)-(3-aminopiperidin-1-yl) (2-(1-(cyclopropylmeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM773981(US20250302842, Example 76)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637618((R)-(3-aminopiperidin-1-yl)(2-(1-(4-fluorobenzyl)-...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637615((R)-(3-aminopiperidin-1-yl)(2-(1-(4-chlorobenzyl)-...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637624((R)-(3-aminopiperidin-1-yl)(2-(1-benzyl-1H-indol-2...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637622((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmethy...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637620((R)-(3-aminopiperidin-1-yl)(2-(1-(pyridin-3-ylmeth...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637606((R)-(3-aminopiperidin-1-yl)(2-(1-ethyl-1H-pyrrolo[...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637661((R)-(3-aminopiperidin-1-yl)(2-(1-(pyridin-3-ylmeth...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637604(((R)-(3-aminopiperidin-1-yl)(2-(1-(cyclopropylmeth...)
Affinity DataIC50: 5.50E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM637605((2-(aminomethyl)piperidin-1-yl)(2-(1-(cyclopropylm...)
Affinity DataIC50: 1.00E+4nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent