Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 4053
TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73108BDBM73108(US20250381168, Example C1)
Affinity DataIC50: 1.10nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73110BDBM73110(US20250381168, Example C17)
Affinity DataIC50: 1.5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73105BDBM73105(US20250381168, Example 9)
Affinity DataIC50: 1.60nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73107BDBM73107(US20250381168, Example 10)
Affinity DataIC50: 3.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73109BDBM73109(US20250381168, Example C6)
Affinity DataIC50: 3.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73104BDBM73104((2S)-2-[[(2S)-1-(3,5-dichlorophenyl)sulfonylpyrrol...)
Affinity DataIC50: 4.80nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73103BDBM73103((2S)-2-[[(2S)-1-(3,5-dichlorophenyl)sulfonylpyrrol...)
Affinity DataIC50: 5.40nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73102BDBM73102(US20250381168, Example 1)
Affinity DataIC50: 5.60nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent

TargetIntegrin alpha-4/beta-7(Human)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 73111BDBM73111(US20250381168, Example BIO5192)
Affinity DataIC50: 1.00E+4nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2026
Entry Details
US Patent