Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 4402
TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496348BDBM50496348(CHEMBL3126185 | US20260007675, Compound 11)
Affinity DataIC50: 390nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496336BDBM50496336(CHEMBL3126186 | US20260007675, Compound 12)
Affinity DataIC50: 1.70E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496343BDBM50496343(CHEMBL3126184 | US20260007675, Compound 10)
Affinity DataIC50: 4.00E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496353BDBM50496353(CHEMBL3126183 | US20260007675, Compound 9)
Affinity DataIC50: 4.10E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496350BDBM50496350(CHEMBL3126202 | US20260007675, Compound 2)
Affinity DataIC50: 1.08E+4nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496337BDBM50496337(CHEMBL3126182 | US20260007675, Compound 8)
Affinity DataIC50: 1.12E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496342BDBM50496342(CHEMBL1438422 | US20260007675, Compound 1)
Affinity DataIC50: 1.28E+4nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496338BDBM50496338(CHEMBL3126181 | US20260007675, Compound 7)
Affinity DataIC50: 1.53E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496352BDBM50496352(CHEMBL3126203 | US20260007675, Compound 3)
Affinity DataIC50: 2.05E+5nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496344BDBM50496344(CHEMBL3126179 | US20260007675, Compound 5)
Affinity DataIC50: 2.34E+5nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496339BDBM50496339(CHEMBL17345 | US20260007675, Compound 4)
Affinity DataIC50: 2.50E+5nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A/Menin(Human)
Memorial Sloan Kettering Cancer Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50496349BDBM50496349(CHEMBL3126180 | US20260007675, Compound 6)
Affinity DataIC50: 2.95E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent