Compile Data Set for Download or QSAR
Report error Found 416 Enz. Inhib. hit(s) with all data for entry = 13506
TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800431BDBM800431(3-(((2-chloro-[1,1'-biphenyl]-4-yl)methyl)amino)-N...)
Affinity DataIC50: 0.190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800432BDBM800432(3-(((2-chloro- [1,1'-biphenyl]- 4- yl)methyl)amino...)
Affinity DataIC50: 0.25nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800464BDBM800464(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 0.280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800483BDBM800483(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 0.280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800436BDBM800436(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol- 4- ...)
Affinity DataIC50: 0.290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800456BDBM800456(3-((3-chloro-4-(trifluoromethoxy)benzyl)amino)-N-(...)
Affinity DataIC50: 0.320nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800478BDBM800478(N-(2-(4-(((5-cyclobutoxy-1H-indol-2-yl)methyl)amin...)
Affinity DataIC50: 0.330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800504BDBM800504(N-(3-((6-(2H- tetrazol-5-yl)- 1H-indazol-4- yl)ami...)
Affinity DataIC50: 0.330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800620BDBM800620((S)-5-(4-((2- ((4-((3-(oxazol- 5-ylmethyl)-5- (tri...)
Affinity DataIC50: 0.410nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800450BDBM800450(N-(3-((6-(2H- 1,2,3-triazol-4- yl)-1H-indazol- 4- ...)
Affinity DataIC50: 0.440nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800474BDBM800474(6-(4H-1,2,4-triazol-4-yl)-N-(2-(4-(((5-(trifluorom...)
Affinity DataIC50: 0.440nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800457BDBM800457(N-(3-((6-(1,2,3-thiadiazol-5-yl)-1H-indazol-4-yl)a...)
Affinity DataIC50: 0.470nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800458BDBM800458(N-(3-((6-(4H-1,2,4-triazol-4-yl)-1H-indazol-4-yl)a...)
Affinity DataIC50: 0.480nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800613BDBM800613(N-(3-((6-(6- aminopyridazin- 4-yl)-1H-indazol- 4- ...)
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800463BDBM800463(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 0.530nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800453BDBM800453(3-(((2-chloro- [1,1'-biphenyl]- 4- yl)methyl)amino...)
Affinity DataIC50: 0.540nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800616BDBM800616(3-((3-chloro-4-(trifluoromethoxy)benzyl)amino)-N-(...)
Affinity DataIC50: 0.570nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800466BDBM800466(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol- 4- ...)
Affinity DataIC50: 0.580nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800437BDBM800437(N-(6-(4H-1,2,4-triazol-4-yl)-1H-indazol-4-yl)-3-(3...)
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800482BDBM800482(N-(2-(4-(((5-cyclobutoxy-1H-indol-2-yl)methyl)amin...)
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800468BDBM800468(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 0.620nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800433BDBM800433(3-(((2-chloro-[1,1'-biphenyl]-4-yl)methyl)amino)-N...)
Affinity DataIC50: 0.620nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800581BDBM800581(3-((3-chloro-4-(trifluoromethoxy)benzyl)amino)-N-(...)
Affinity DataIC50: 0.640nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800593BDBM800593(3-((3-chloro-4- (trifluoromethoxy) benzyl)amino)- ...)
Affinity DataIC50: 0.640nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800497BDBM800497(N1-(2-((6-(4H-1,2,4-triazol-4-yl)-1H-indazol-4-yl)...)
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800476BDBM800476(N-(2-(4-(((1- methyl-5- (trifluoromethyl)- 1H-indo...)
Affinity DataIC50: 0.710nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800610BDBM800610(3-((3-chloro-4-(trifluoromethoxy)benzyl)amino)-N-(...)
Affinity DataIC50: 0.760nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800619BDBM800619((S)-2-(3-(((5- (2-((6-(6- hydroxypyrida- zin-4-yl)...)
Affinity DataIC50: 0.760nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800428BDBM800428(N-(3-((6-(1H- pyrazol-4-yl)- 1H-indazol-4- yl)amin...)
Affinity DataIC50: 0.770nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800518BDBM800518(6-(pyridazin-4- yl)-N-(2-(4-(((5- (trifluoromethyl...)
Affinity DataIC50: 0.770nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800462BDBM800462(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 0.780nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800449BDBM800449(N1-(2-((6-(4H-1,2,4-triazol-4-yl)-1H-indazol-4-yl)...)
Affinity DataIC50: 0.780nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800523BDBM800523(N-(2-(4-(((5- cyclobutoxy-1H- indol-2-yl)methyl)am...)
Affinity DataIC50: 0.820nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800543BDBM800543(4-(2-((6-(4H- 1,2,4-triazol-4-yl)-1H- indazol-4-yl...)
Affinity DataIC50: 0.860nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800626BDBM800626(3-(4-((2-(4-((3,5-difluoro-4-(trifluoromethoxy)ben...)
Affinity DataIC50: 0.870nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800500BDBM800500(3-(((2-chloro- [1,1'-biphenyl]- 4- yl)methyl)amino...)
Affinity DataIC50: 0.890nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800609BDBM800609(N-(3-((6-(2- aminopyridin- 4-yl)-1H- indazol-4- yl...)
Affinity DataIC50: 0.940nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800452BDBM800452(3-(((2-chloro- [1,1'-biphenyl]- 4- yl)methyl)amino...)
Affinity DataIC50: 0.950nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800470BDBM800470(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 0.950nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800455BDBM800455(4-(4-((3-(3- (((2-chloro- [1,1'-biphenyl]- 4- yl)m...)
Affinity DataIC50: 0.990nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800598BDBM800598(N-(3-((6-(1,2,4-oxadiazol-5-yl)-1H-indazol-4-yl)am...)
Affinity DataIC50: 1.17nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800618BDBM800618((S)-5-(4-((2-((4-((3-(hydroxymethyl)-5-(trifluorom...)
Affinity DataIC50: 1.21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800480BDBM800480(N-((5-cyclobutoxy-1H- indol-2-yl)methyl)- 4-(2-((6...)
Affinity DataIC50: 1.25nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800447BDBM800447(3-(((2-Chloro- [1,1'-biphenyl]- 4- yl)methyl)amino...)
Affinity DataIC50: 1.35nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800496BDBM800496(3-(((2-chloro-[1,1'-biphenyl]-4-yl)methyl)amino)-N...)
Affinity DataIC50: 1.37nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800426BDBM800426(3-(((2-Chloro-[1,1'-biphenyl]-4-yl)methyl)amino)-N...)
Affinity DataIC50: 1.38nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800461BDBM800461(N-(3-((6-(4H- 1,2,4-triazol-4- yl)-1H-indazol-4- y...)
Affinity DataIC50: 1.39nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800522BDBM800522(6-(isoxazol-4- yl)-N-(2-(4-(((5- (trifluoromethyl)...)
Affinity DataIC50: 1.42nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800477BDBM800477(N-(2-(4-(((6- chloro-1H- indol-2- yl)methyl)amino)...)
Affinity DataIC50: 1.43nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha(Human)
Cambridge Enterprise

US Patent
LigandChemical structure of BindingDB Monomer ID 800438BDBM800438(N-(3-((6-(4H-1,2,4-triazol-4-yl)-1H-indazol-4-yl)a...)
Affinity DataIC50: 1.43nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/5/2026
Entry Details
US Patent

Displayed 1 to 50 (of 416 total ) | Next | Last >>
Jump to: