Compile Data Set for Download or QSAR
Report error Found 185 Enz. Inhib. hit(s) with all data for entry = 5879
TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98187BDBM98187(US8486940, 89 | US9650362, 89)
Affinity DataKi:  12.5nM IC50: 160nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98186BDBM98186(US8486940, 73 | US9650362, 73)
Affinity DataKi:  33.6nM IC50: 170nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98182BDBM98182(US8486940, 14)
Affinity DataKi:  37.4nM IC50: 238nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98183BDBM98183(US8486940, 43)
Affinity DataKi:  40.8nM IC50: 254nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98188BDBM98188(US8486940, 142)
Affinity DataKi:  53.5nM IC50: 297nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98189BDBM98189(US8486940, 145)
Affinity DataKi:  58.8nM IC50: 240nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98180BDBM98180(US8486940, 12)
Affinity DataKi:  62.5nM IC50: 482nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98184BDBM98184(US8486940, 55)
Affinity DataKi:  75nM IC50: 397nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98185BDBM98185(US8486940, 60 | US9650362, 60)
Affinity DataKi:  149nM IC50: 882nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 98181BDBM98181(US8486940, 13)
Affinity DataKi:  7.25E+3nM IC50: 3.02E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65023BDBM65023(US8486940, 225)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65024BDBM65024(US8486940, 226)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65025BDBM65025(US8486940, 227)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65026BDBM65026(US8486940, 228)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65018BDBM65018(US8486940, 219)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65019BDBM65019(US8486940, 220)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65021BDBM65021(US8486940, 221)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65022BDBM65022(US8486940, 224)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65027BDBM65027(US8486940, 232)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65028BDBM65028(US8486940, 233)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 65029BDBM65029(US8486940, 234)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64588BDBM64588(US8486940, 2)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64590BDBM64590(US8486940, 3)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64592BDBM64592(US8486940, 7 | US8486940, 5)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64602BDBM64602(US8486940, 11)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64606BDBM64606(US8486940, 15)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64607BDBM64607(US8486940, 16)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64609BDBM64609(US8486940, 17)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64592BDBM64592(US8486940, 7 | US8486940, 5)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64594BDBM64594(US8486940, 8)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64599BDBM64599(US8486940, 9)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64601BDBM64601(US8486940, 10)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64614BDBM64614(US8486940, 22)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64615BDBM64615(US8486940, 23)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64617BDBM64617(US8486940, 24)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64620BDBM64620(US8486940, 25)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64610BDBM64610(US8486940, 18)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64611BDBM64611(US8486940, 19)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64612BDBM64612(US8486940, 20)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64613BDBM64613(US8486940, 21)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64629BDBM64629(US8486940, 30)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64630BDBM64630(US8486940, 32)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64631BDBM64631(US8486940, 33)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64632BDBM64632(US8486940, 34)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64621BDBM64621(US8486940, 26)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64622BDBM64622(US8486940, 27)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64624BDBM64624(US8486940, 28)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64628BDBM64628(US8486940, 29)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64640BDBM64640(US8486940, 39)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 64642BDBM64642(US8486940, 40)
Affinity DataIC50: 1.00E+4nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2013
Entry Details
US Patent

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