Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 5873
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98040(US8486953, 53)
Affinity DataIC50:  6nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98034(US8486953, 9)
Affinity DataIC50:  27nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98032(US8486953, 2)
Affinity DataIC50:  28nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98035(US8486953, 10)
Affinity DataIC50:  34nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98040(US8486953, 53)
Affinity DataIC50:  35nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98033(US8486953, 6)
Affinity DataIC50:  35nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98036(US8486953, 19)
Affinity DataIC50:  60nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98039(US8486953, 48)
Affinity DataIC50:  92nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98034(US8486953, 9)
Affinity DataIC50:  100nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98038(US8486953, 41)
Affinity DataIC50:  110nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98032(US8486953, 2)
Affinity DataIC50:  120nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98041(US8486953, 71)
Affinity DataIC50:  160nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98033(US8486953, 6)
Affinity DataIC50:  180nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98038(US8486953, 41)
Affinity DataIC50:  210nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98035(US8486953, 10)
Affinity DataIC50:  210nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98041(US8486953, 71)
Affinity DataIC50:  400nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98039(US8486953, 48)
Affinity DataIC50:  460nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98037(US8486953, 34)
Affinity DataIC50:  560nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98036(US8486953, 19)
Affinity DataIC50:  590nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM98037(US8486953, 34)
Affinity DataIC50:  680nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent