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Found 52 Enz. Inhib. hit(s) with all data for entry = 5907
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99943(US8501750, 56)
Affinity DataIC50:  0.340nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99950(US8501750, 83)
Affinity DataIC50:  0.770nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99946(US8501750, 60)
Affinity DataIC50:  1nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99949(US8501750, 76)
Affinity DataIC50:  1nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99952(US8501750, 105)
Affinity DataIC50:  1nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99953(US8501750, 107)
Affinity DataIC50:  1.10nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99947(US8501750, 63)
Affinity DataIC50:  1.10nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99981(US8501750, 186)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99980(US8501750, 181)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99961(US8501750, 131)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99951(US8501750, 99)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99945(US8501750, 59)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99992(US8501750, 215)
Affinity DataIC50:  1.30nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99974(US8501750, 153)
Affinity DataIC50:  1.30nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99958(US8501750, 127)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99993(US8501750, 221)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99954(US8501750, 109)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99984(US8501750, 197)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99977(US8501750, 157)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99988(US8501750, 209)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99967(US8501750, 143)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99964(US8501750, 136)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99985(US8501750, 198)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99963(US8501750, 135)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99966(US8501750, 142)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99972(US8501750, 150)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99948(US8501750, 73)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99970(US8501750, 148)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99987(US8501750, 205)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99973(US8501750, 152)
Affinity DataIC50:  1.5nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99959(US8501750, 129)
Affinity DataIC50:  1.60nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99944(US8501750, 58)
Affinity DataIC50:  1.60nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99979(US8501750, 180)
Affinity DataIC50:  1.60nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99960(US8501750, 130)
Affinity DataIC50:  1.60nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99995(US8501750, 225)
Affinity DataIC50:  1.60nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99989(US8501750, 210)
Affinity DataIC50:  1.60nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99983(US8501750, 194)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99978(US8501750, 158)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99969(US8501750, 145)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99965(US8501750, 140)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99962(US8501750, 132)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99957(US8501750, 121)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99968(US8501750, 144)
Affinity DataIC50:  1.70nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99991(US8501750, 214)
Affinity DataIC50:  1.80nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99955(US8501750, 116)
Affinity DataIC50:  1.80nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99956(US8501750, 117)
Affinity DataIC50:  1.80nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99986(US8501750, 203)
Affinity DataIC50:  1.80nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99971(US8501750, 149)
Affinity DataIC50:  1.80nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99994(US8501750, 222)
Affinity DataIC50:  1.90nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99976(US8501750, 154)
Affinity DataIC50:  1.90nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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