Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 5901
TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99498(US8501768, 26)
Affinity DataIC50: 33nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99474(US8501768, 2)
Affinity DataIC50: 49.5nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99483(US8501768, 11)
Affinity DataIC50: 50.1nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99489(US8501768, 17)
Affinity DataIC50: 51.2nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99505(US8501768, 33)
Affinity DataIC50: 96.5nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99477(US8501768, 5)
Affinity DataIC50: 136nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99508(US8501768, 36)
Affinity DataIC50: 139nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99496(US8501768, 24)
Affinity DataIC50: 153nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99495(US8501768, 23)
Affinity DataIC50: 161nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99473(US8501768, 1)
Affinity DataIC50: 170nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99485(US8501768, 13)
Affinity DataIC50: 174nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99490(US8501768, 18)
Affinity DataIC50: 244nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99480(US8501768, 8)
Affinity DataIC50: 259nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99492(US8501768, 20)
Affinity DataIC50: 268nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99504(US8501768, 32)
Affinity DataIC50: 279nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99479(US8501768, 7)
Affinity DataIC50: 311nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99493(US8501768, 21)
Affinity DataIC50: 327nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99497(US8501768, 25)
Affinity DataIC50: 334nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99475(US8501768, 3)
Affinity DataIC50: 354nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99478(US8501768, 6)
Affinity DataIC50: 359nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99484(US8501768, 12)
Affinity DataIC50: 380nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99481(US8501768, 9)
Affinity DataIC50: 438nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99503(US8501768, 31)
Affinity DataIC50: 443nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99506(US8501768, 34)
Affinity DataIC50: 482nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99502(US8501768, 30)
Affinity DataIC50: 502nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99507(US8501768, 35)
Affinity DataIC50: 554nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99501(US8501768, 29)
Affinity DataIC50: 637nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99499(US8501768, 27)
Affinity DataIC50: 700nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99494(US8501768, 22)
Affinity DataIC50: 701nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99476(US8501768, 4)
Affinity DataIC50: 710nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99487(US8501768, 15)
Affinity DataIC50: 727nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99486(US8501768, 14)
Affinity DataIC50: 845nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99491(US8501768, 19)
Affinity DataIC50: 867nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99500(US8501768, 28)
Affinity DataIC50: 896nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99488(US8501768, 16)
Affinity DataIC50: 953nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent

TargetHormone-sensitive lipase(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM99482(US8501768, 10)
Affinity DataIC50: 956nMAssay Description:HSL enzyme activity was measured by a colorimetric assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2013
Entry Details
US Patent