Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 5924
TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100778BDBM100778(US8507535, 17)
Affinity DataKi:  2.30nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100777BDBM100777(US8507535, 16)
Affinity DataKi:  3.70nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100768BDBM100768(US8507535, 7)
Affinity DataKi:  4.30nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100786BDBM100786(US8507535, 25)
Affinity DataKi:  4.40nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100779BDBM100779(US8507535, 18)
Affinity DataKi:  5.90nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100764BDBM100764(US8507535, 3)
Affinity DataKi:  7.20nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100774BDBM100774(US8507535, 13)
Affinity DataKi:  8.70nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100772BDBM100772(US8507535, 11)
Affinity DataKi:  10.6nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100780BDBM100780(US8507535, 19)
Affinity DataKi:  11.2nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100787BDBM100787(US8507535, 26)
Affinity DataKi:  11.4nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100776BDBM100776(US8507535, 15)
Affinity DataKi:  15nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100775BDBM100775(US8507535, 14)
Affinity DataKi:  15nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100781BDBM100781(US8507535, 20)
Affinity DataKi:  19.3nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100773BDBM100773(US8507535, 12)
Affinity DataKi:  22.5nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100762BDBM100762(US8507535, 1)
Affinity DataKi:  24.2nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100785BDBM100785(US8507535, 24)
Affinity DataKi:  26.1nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100783BDBM100783(US8507535, 22)
Affinity DataKi:  27.2nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100767BDBM100767(US8507535, 6)
Affinity DataKi:  35.2nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100782BDBM100782(US8507535, 21)
Affinity DataKi:  39nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100769BDBM100769(US8507535, 8)
Affinity DataKi:  45.1nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100763BDBM100763(US8507535, 2)
Affinity DataKi:  47.8nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100770BDBM100770(US8507535, 9)
Affinity DataKi:  56.3nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100766BDBM100766(US8507535, 5)
Affinity DataKi:  61.8nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100771BDBM100771(US8507535, 10)
Affinity DataKi:  87.4nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 100788BDBM100788(US8507535, 27)
Affinity DataKi:  93.1nMAssay Description:Competition binding assay using hNK3 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2013
Entry Details
US Patent