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Found 11 Enz. Inhib. hit(s) with all data for entry = 6034
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104989(US8569291, 11 | US8569291, 12)
Affinity DataKi:  0.210nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104991(US8569291, 13)
Affinity DataKi:  1.60nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104979(US8569291, 1)
Affinity DataKi:  25nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104989(US8569291, 11 | US8569291, 12)
Affinity DataKi:  29nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104985(US8569291, 7)
Affinity DataKi:  35nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104986(US8569291, 8)
Affinity DataKi:  130nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104987(US8569291, 9)
Affinity DataKi:  160nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104980(US8569291, 2)
Affinity DataKi:  570nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104984(US8569291, 6)
Affinity DataKi:  630nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104981(US8569291, 3)
Affinity DataKi:  2.60E+3nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM104982(US8569291, 4)
Affinity DataKi:  6.40E+3nMAssay Description:Recombinant receptor binding assay using human CL receptor/RAMP1 (CGRP).More data for this Ligand-Target Pair
In DepthDetails US Patent