Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 6567
TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139462BDBM139462(US8614195, 4)
Affinity DataIC50: 2.40nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139452BDBM139452(US8614195, 2)
Affinity DataIC50: 17.5nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139463BDBM139463(US8614195, 1)
Affinity DataIC50: 22.5nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139456BDBM139456(US8614195, 2c)
Affinity DataIC50: 27nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139452BDBM139452(US8614195, 2)
Affinity DataIC50: 35nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139457BDBM139457(US8614195, 2e)
Affinity DataIC50: 89nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139462BDBM139462(US8614195, 4)
Affinity DataIC50: 89.3nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139454BDBM139454(US8614195, 2a)
Affinity DataIC50: 97nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139458BDBM139458(US8614195, 2f)
Affinity DataIC50: 143nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139455BDBM139455(US8614195, 2b)
Affinity DataIC50: 186nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139457BDBM139457(US8614195, 2e)
Affinity DataIC50: 188nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139456BDBM139456(US8614195, 2c)
Affinity DataIC50: 197nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139454BDBM139454(US8614195, 2a)
Affinity DataIC50: 308nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139455BDBM139455(US8614195, 2b)
Affinity DataIC50: 338nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139463BDBM139463(US8614195, 1)
Affinity DataIC50: 409nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139459BDBM139459(US8614195, 2g)
Affinity DataIC50: 567nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139460BDBM139460(US8614195, 3)
Affinity DataIC50: 814nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139460BDBM139460(US8614195, 3)
Affinity DataIC50: 1.00E+3nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139461BDBM139461(US8614195, 3a)
Affinity DataIC50: 1.00E+3nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139459BDBM139459(US8614195, 2g)
Affinity DataIC50: 1.00E+3nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139458BDBM139458(US8614195, 2f)
Affinity DataIC50: 3.44E+3nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetSodium/glucose cotransporter 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 139461BDBM139461(US8614195, 3a)
Affinity DataIC50: 5.65E+3nMAssay Description:The ability of the substances to inhibit the SGLT-2 activity may be demonstrated in a test set-up in which a CHO-K1 cell line (ATCC No. CCL 6 1) or a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent