Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 6288
TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120757BDBM120757(US8703761, 1-29)
Affinity DataIC50: 3.5nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120755BDBM120755(US8703761, 1-8)
Affinity DataIC50: 8.5nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120756BDBM120756(US8703761, 1-28)
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120759BDBM120759(US8703761, 8-1)
Affinity DataIC50: 54.5nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120753BDBM120753(US8703761, 1-1)
Affinity DataIC50: 60.5nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120758BDBM120758(US8703761, 6-14)
Affinity DataIC50: 197nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120763BDBM120763(US8703761, 14-4)
Affinity DataIC50: 225nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120760BDBM120760(US8703761, 8-2)
Affinity DataIC50: 240nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120754BDBM120754(US8703761, 1-6)
Affinity DataIC50: 241nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120767BDBM120767(US8703761, 6-1)
Affinity DataIC50: 910nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120761BDBM120761(US8703761, 12-3)
Affinity DataIC50: 1.18E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120765BDBM120765(US8703761, 14-24)
Affinity DataIC50: 1.75E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120762BDBM120762(US8703761, 12-4)
Affinity DataIC50: 2.08E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120764BDBM120764(US8703761, 14-3)
Affinity DataIC50: 2.30E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent

TargetDiacylglycerol O-acyltransferase 1 [89-488](Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 120766BDBM120766(US8703761, 14-28)
Affinity DataIC50: 6.13E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
US Patent