Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 6331
TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123511BDBM123511(US8748435, 36)
Affinity DataIC50: 5nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123488BDBM123488(US8748435, 13)
Affinity DataIC50: 7nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123489BDBM123489(US8748435, 14)
Affinity DataIC50: 10nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123514BDBM123514(US8748435, 39)
Affinity DataIC50: 13nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123480BDBM123480(US8748435, 5)
Affinity DataIC50: 15nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123513BDBM123513(US8748435, 38)
Affinity DataIC50: 15nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123497BDBM123497(US8748435, 22)
Affinity DataIC50: 19nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123484BDBM123484(US8748435, 9)
Affinity DataIC50: 19nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123504BDBM123504(US8748435, 29)
Affinity DataIC50: 21nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123496BDBM123496(US8748435, 21)
Affinity DataIC50: 22nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123481BDBM123481(US8748435, 6)
Affinity DataIC50: 24nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123505BDBM123505(US8748435, 30)
Affinity DataIC50: 26nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123483BDBM123483(US8748435, 8)
Affinity DataIC50: 28nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123492BDBM123492(US8748435, 17)
Affinity DataIC50: 30nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123485BDBM123485(US8748435, 10)
Affinity DataIC50: 33nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123487BDBM123487(US8748435, 12)
Affinity DataIC50: 33nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123482BDBM123482(US8748435, 7)
Affinity DataIC50: 34nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123477BDBM123477(US8748435, 2)
Affinity DataIC50: 34nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123498BDBM123498(US8748435, 23)
Affinity DataIC50: 35nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123491BDBM123491(US8748435, 16)
Affinity DataIC50: 35nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123486BDBM123486(US8748435, 11)
Affinity DataIC50: 38nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123508BDBM123508(US8748435, 33)
Affinity DataIC50: 38nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123506BDBM123506(US8748435, 31)
Affinity DataIC50: 43nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123501BDBM123501(US8748435, 26)
Affinity DataIC50: 44nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123478BDBM123478(US8748435, 3)
Affinity DataIC50: 44nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123476BDBM123476(US8748435, 1)
Affinity DataIC50: 45nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123479BDBM123479(US8748435, 4)
Affinity DataIC50: 47nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123490BDBM123490(US8748435, 15)
Affinity DataIC50: 51nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123499BDBM123499(US8748435, 24)
Affinity DataIC50: 54nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123494BDBM123494(US8748435, 19)
Affinity DataIC50: 54nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123515BDBM123515(US8748435, 40)
Affinity DataIC50: 55nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123502BDBM123502(US8748435, 27)
Affinity DataIC50: 59nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123510BDBM123510(US8748435, 35)
Affinity DataIC50: 74nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123509BDBM123509(US8748435, 34)
Affinity DataIC50: 77nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123493BDBM123493(US8748435, 18)
Affinity DataIC50: 81nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123500BDBM123500(US8748435, 25)
Affinity DataIC50: 110nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent

TargetG-protein coupled receptor 4(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 123503BDBM123503(US8748435, 28)
Affinity DataIC50: 118nMpH: 8.0Assay Description:Serial dilutions of compounds (stock in 10 mM DMSO) are prepared by first diluting the compounds in DMSO followed by a 1:50 dilution into assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
US Patent