Compile Data Set for Download or QSAR
Report error Found 151 Enz. Inhib. hit(s) with all data for entry = 6349
TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123945BDBM123945(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 7nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123951BDBM123951(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 10nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124052BDBM124052(US8754233, 5-(3-Amino-propyl)-4-benzothiazol-2-yl-...)
Affinity DataIC50: 10nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124022BDBM124022(US8754233, 4-Benzothiazol-2-yl-5-(3-methylamino-pr...)
Affinity DataIC50: 20nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124067BDBM124067(US8754233, N3-(2-Amino-ethyl)-4-benzothiazol-2-yl-...)
Affinity DataIC50: 20nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123930BDBM123930(US8754233, 2-(3-Amino-1H-pyrazol-4-yl)-5-fluoro-be...)
Affinity DataIC50: 20nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123965BDBM123965(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 40nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123933BDBM123933(US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 40nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124001BDBM124001(US8754233, 4-(5-Fluoro-benzothiazol-2-yl)-5-methyl...)
Affinity DataIC50: 40nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123943BDBM123943(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-4-...)
Affinity DataIC50: 40nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123992BDBM123992(US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...)
Affinity DataIC50: 40nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123969BDBM123969(US8754233, 2-(5-Amino-3-pyridin-4-yl-1H-pyrazol-4-...)
Affinity DataIC50: 50nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123999BDBM123999(US8754233, 4-(5-Fluoro-6-methyl-benzothiazol-2-yl)...)
Affinity DataIC50: 50nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123946BDBM123946(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 50nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124033BDBM124033(US8754233, 4-Benzothiazol-2-yl-5-piperidin-4-yl-2H...)
Affinity DataIC50: 60nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123942BDBM123942(US8754233, 2-(5-Amino-1H-pyrazol-4-yl)-benzothiazo...)
Affinity DataIC50: 60nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123932BDBM123932(US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 60nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123994BDBM123994(US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...)
Affinity DataIC50: 60nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123936BDBM123936(US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 70nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123996BDBM123996(US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...)
Affinity DataIC50: 70nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123931BDBM123931(US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-4,...)
Affinity DataIC50: 70nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123962BDBM123962(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 90nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124028BDBM124028(US8754233, 4-Benzothiazol-2-yl-5-furan-2-yl-2H-pyr...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124053BDBM124053(US8754233, 5-(4-Amino-phenyl)-4-benzothiazol-2-yl-...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123925BDBM123925(US8754233, [2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123972BDBM123972(US8754233, 2-{[2-(5-Amino-3-methyl-1H-pyrazol-4-yl...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124035BDBM124035(US8754233, 4-Benzothiazol-2-yl-5-pyridin-4-yl-2H-p...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123993BDBM123993(US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124024BDBM124024(US8754233, 4-Benzothiazol-2-yl-5-(4-methylamino-bu...)
Affinity DataIC50: 100nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123947BDBM123947(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 130nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123944BDBM123944(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 150nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124041BDBM124041(US8754233, 4-Benzothiazol-2-yl-N3-(2-ethylamino-et...)
Affinity DataIC50: 150nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124032BDBM124032(US8754233, 4-Benzothiazol-2-yl-5-piperazin-1-yl-2H...)
Affinity DataIC50: 190nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123998BDBM123998(US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123997BDBM123997(US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124069BDBM124069(US8754233, N3-(3-Dimethylamino-propyl)-4-(5-fluoro...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123973BDBM123973(US8754233, 3-(5-Amino-4-benzothiazol-2-yl-1H-pyraz...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124004BDBM124004(US8754233, 4-(6-Bromo-5-fluoro-benzothiazol-2-yl)-...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123948BDBM123948(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124009BDBM124009(US8754233, 4-(6-Fluoro-benzothiazol-2-yl)-1H-pyraz...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124008BDBM124008(US8754233, 4-(6-Dimethylaminomethyl-benzothiazol-2...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123952BDBM123952(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124013BDBM124013(US8754233, 4-(6-Methoxy-benzothiazol-2-yl)-5-piper...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123923BDBM123923(US8754233, (4-Benzothiazol-2-yl-1H-pyrazol-3-yl)-[...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123960BDBM123960(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124021BDBM124021(US8754233, 4-Benzothiazol-2-yl-5-(3-dimethylamino-...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123963BDBM123963(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 124055BDBM124055(US8754233, 5-Methyl-4-(4,5,6-trifluoro-benzothiazo...)
Affinity DataIC50: 200nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123935BDBM123935(US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 300nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetIntegrin-linked protein kinase(Human)
Dermira (Canada)

US Patent
LigandChemical structure of BindingDB Monomer ID 123966BDBM123966(US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...)
Affinity DataIC50: 300nMT: 2°CAssay Description:5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

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