Compile Data Set for Download or QSAR
Report error Found 162 Enz. Inhib. hit(s) with all data for entry = 6366
LigandChemical structure of BindingDB Monomer ID 50403100BDBM50403100(CHEMBL2216891 | US8765940, 4-(3,3-dimethyl-6-(4-mo...)
Affinity DataKi:  1.05nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124797BDBM124797(US8765940, 1-(5,7-difluoro-3-methyl-4-(6'-(4-morph...)
Affinity DataKi:  1.27nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124781BDBM124781(US8765940, 1-(7-fluoro-3-methyl-2-(2-pyridinyl)-4-...)
Affinity DataKi:  1.37nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124778BDBM124778(US8765940, 1-(5,7-difluoro-3-methyl-4-(6'-(4-m...)
Affinity DataKi:  1.49nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124765BDBM124765(US8765940, 1'-(5,7-difluoro-3-methyl-2-(5-meth...)
Affinity DataKi:  1.51nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124764BDBM124764(US8765940, 2-(2,2-dimethyl-4-morpholinyl)-4-(3,3-d...)
Affinity DataKi:  1.52nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124749BDBM124749(US8765940, 1-(4-(3,3-dimethyl-6-(4-morpholinyl)-2,...)
Affinity DataKi:  1.54nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124759BDBM124759(US8765940, 1-(7-fluoro-3-methyl-4-(6'-(4-morph...)
Affinity DataKi:  1.62nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124767BDBM124767(US8765940, 1-(7-fluoro-3-methyl-2-(4-methyl-2-pyri...)
Affinity DataKi:  1.96nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124766BDBM124766(US8765940, 1-(7-fluoro-3-methyl-2-(2-pyridinyl)-4-...)
Affinity DataKi:  2.22nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124799BDBM124799(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.24nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124798BDBM124798(US8765940, 1-(5,7-difluoro-3-methyl-4-(6'-(4-morph...)
Affinity DataKi:  2.30nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124783BDBM124783(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.30nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124743BDBM124743(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.34nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124758BDBM124758(US8765940, 1-(5,7-difluoro-3-methyl-4-(6'-(4-morph...)
Affinity DataKi:  2.36nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124775BDBM124775(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.36nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124676BDBM124676(US8765940, 4-(1-(7-fluoro-3-methyl-2-(2-(methylsul...)
Affinity DataKi:  2.44nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124734BDBM124734(US8765940, 3-((4-(3,3-dimethyl-6-(4-morpholinyl)-2...)
Affinity DataKi:  2.68nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124757BDBM124757(US8765940, 1'-(8-chloro-2,3-dimethyl-4-quinoli...)
Affinity DataKi:  2.68nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124779BDBM124779(US8765940, tert-butyl 4-(5,7-difluoro-3-methyl-4-(...)
Affinity DataKi:  2.70nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124731BDBM124731(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.77nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124732BDBM124732(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.87nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124728BDBM124728(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  2.90nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124747BDBM124747(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  3nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124777BDBM124777(US8765940, methyl 4-(5,7-difluoro-3-methyl-4-(6...)
Affinity DataKi:  3.11nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124742BDBM124742(US8765940, 1-(4-(3,3-dimethyl-6-(4-morpholinyl)-2,...)
Affinity DataKi:  3.14nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124796BDBM124796(US8765940, 4-(5,7-difluoro-3-methyl-4-(6'-(4-morph...)
Affinity DataKi:  3.16nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124727BDBM124727(US8765940, 2-benzyl-4-(3,3-dimethyl-6-(4-morpholin...)
Affinity DataKi:  3.20nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50396616BDBM50396616(CHEMBL2171930 | US8765940, 4-(1-(7-fluoro-3-methyl...)
Affinity DataKi:  3.32nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124683BDBM124683(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  3.33nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124667BDBM124667(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  4.07nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124688BDBM124688(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  4.07nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124741BDBM124741(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  4.17nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124786BDBM124786(US8765940, 1'-(3-methyl-2-phenyl-1,8-naphthyri...)
Affinity DataKi:  4.36nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124675BDBM124675(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  4.43nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124755BDBM124755(US8765940, 1'-(5,7-difluoro-3-methyl-2-(2-(met...)
Affinity DataKi:  4.51nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124756BDBM124756(US8765940, 1-(5,7-difluoro-3-methyl-4-(6-(4-morpho...)
Affinity DataKi:  4.64nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124761BDBM124761(US8765940, 1'-(7-fluoro-3-methyl-2-(4-methyl-2...)
Affinity DataKi:  5.19nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124746BDBM124746(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  5.21nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124801BDBM124801(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  5.37nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124784BDBM124784(US8765940, 1'-(2-(3-fluorophenyl)-3-methyl-1,8...)
Affinity DataKi:  5.38nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124763BDBM124763(US8765940, 1'-(2-(2,2-dimethyl-4-morpholinyl)-...)
Affinity DataKi:  5.40nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124751BDBM124751(US8765940, 1-(5,7-difluoro-3-methyl-4-(6'-(4-m...)
Affinity DataKi:  5.51nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124665BDBM124665(US8765940, 4-(3,3-dimethyl-6-(4-morpholinyl)-2,3-d...)
Affinity DataKi:  5.87nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124736BDBM124736(US8765940, 4-(6-(3,6-dihydro-2H-pyran-4-yl)-3,3-di...)
Affinity DataKi:  6.47nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124753BDBM124753(US8765940, 1'-(5-fluoro-3-methyl-2-(2-pyridiny...)
Affinity DataKi:  6.48nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50396610BDBM50396610(CHEMBL2171929 | US8765940, 4-(3,3-dimethyl-6-(4-mo...)
Affinity DataKi:  6.76nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124762BDBM124762(US8765940, 1'-(5,7-difluoro-2-(2-methoxy-4-pyr...)
Affinity DataKi:  6.89nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124769BDBM124769(US8765940, 1-(7-fluoro-3-methyl-4-(6'-(4-morpholin...)
Affinity DataKi:  7.64nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50396613BDBM50396613(CHEMBL2171924 | US8765940, 1-(7-fluoro-3-methyl-2-...)
Affinity DataKi:  7.75nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

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