Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 6375
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124974(US8772508, 8)
Affinity DataKi:  11nM IC50: 580nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM50299866(CHEMBL578153 | US8772508, 6 | N-(1-(3-(5-Methyl-1H...)
Affinity DataKi:  34nM IC50: 430nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM50299867(CHEMBL565907 | US8772508, 10 | N-(1-(3-(5-Methyl-1...)
Affinity DataKi:  41nM IC50: 230nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM50299865(US8772508, 7 | CHEMBL567406 | N-(-1-(3-(5-Methyl-1...)
Affinity DataKi:  51nM IC50: 320nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124971(US8772508, 2)
Affinity DataKi:  55nM IC50: 530nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM50299868(US8772508, 5 | CHEMBL565908 | N-(1-(3-(5-Methyl-1H...)
Affinity DataKi:  67nM IC50: 460nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124975(US8772508, 9)
Affinity DataKi:  67nM IC50: 340nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124973(US8772508, 4)
Affinity DataKi:  76nM IC50: 730nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM50299864(US8772508, 1 | CHEMBL574357 | N-(1-(3-(5-Methyl-1H...)
Affinity DataKi:  80nM IC50: 340nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124972(US8772508, 3)
Affinity DataKi:  96nM IC50: 620nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124981(US8772508, 18)
Affinity DataIC50: 7.46E+3nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124976(US8772508, 11)
Affinity DataIC50: 8.60E+3nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124977(US8772508, 14)
Affinity DataIC50: 8.73E+3nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM50299852(CHEMBL568073 | US8772508, 13 | N-(1-(3-(4-Methyl-1...)
Affinity DataIC50: 8.79E+3nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124979(US8772508, 16)
Affinity DataIC50: 9.45E+3nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124978(US8772508, 15)
Affinity DataIC50: 9.68E+3nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandPNGBDBM124980(US8772508, 17)
Affinity DataIC50: 1.04E+4nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
US Patent