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Found 44 Enz. Inhib. hit(s) with all data for entry = 6418
LigandPNGBDBM20557(AMG 517 | CHEMBL229430 | JMC503515 Compound 23 | N...)
Affinity DataIC50:  20nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128023(US8796328, C)
Affinity DataIC50:  35nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM128033(US8796328, 10)
Affinity DataIC50:  54nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128022(US8796328, B | US8802711, I)
Affinity DataIC50:  55nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM50264258(1-(3-Methylpyridin-2-yl)-N-(4-(trifluoromethylsulf...)
Affinity DataIC50:  100nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128024(US8796328, 1)
Affinity DataIC50:  104nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128032(US8796328, 9)
Affinity DataIC50:  109nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM50321851((R)-8-{5-[3-Methyl-4-(trifluoromethyl)phenyl]oxazo...)
Affinity DataIC50:  180nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128037(US8796328, 14)
Affinity DataIC50:  209nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128057(US8796328, 37)
Affinity DataIC50:  256nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128028(US8796328, 5)
Affinity DataIC50:  325nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128031(US8796328, 8)
Affinity DataIC50:  330nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128058(US8796328, 38)
Affinity DataIC50:  345nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128046(US8796328, 23)
Affinity DataIC50:  358nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128036(US8796328, 13)
Affinity DataIC50:  418nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128042(US8796328, 19)
Affinity DataIC50:  466nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128056(US8796328, 36)
Affinity DataIC50:  587nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128047(US8796328, 25)
Affinity DataIC50:  602nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128059(US8796328, 39)
Affinity DataIC50:  615nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128030(US8796328, 7)
Affinity DataIC50:  747nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128043(US8796328, 20)
Affinity DataIC50:  791nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128038(US8796328, 15)
Affinity DataIC50:  863nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128054(US8796328, 32)
Affinity DataIC50:  913nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128051(US8796328, 29)
Affinity DataIC50:  1.15E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128064(US8796328, 44)
Affinity DataIC50:  1.28E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128026(US8796328, 3)
Affinity DataIC50:  1.81E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128041(US8796328, 18)
Affinity DataIC50:  2.15E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128055(US8796328, 35)
Affinity DataIC50:  2.44E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128029(US8796328, 6)
Affinity DataIC50:  2.90E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128040(US8796328, 17)
Affinity DataIC50:  3.03E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128053(US8796328, 31)
Affinity DataIC50:  3.80E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128061(US8796328, 41)
Affinity DataIC50:  5.28E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128063(US8796328, 43)
Affinity DataIC50:  6.41E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128044(US8796328, 21)
Affinity DataIC50:  7.56E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128045(US8796328, 22)
Affinity DataIC50:  7.59E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128060(US8796328, 40)
Affinity DataIC50:  1.01E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128027(US8796328, 4)
Affinity DataIC50:  1.65E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128049(US8796328, 27)
Affinity DataIC50:  2.25E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128039(US8796328, 16)
Affinity DataIC50:  2.28E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128050(US8796328, 28)
Affinity DataIC50:  2.95E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128062(US8796328, 42)
Affinity DataIC50:  3.28E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM128052(US8796328, 30)
Affinity DataIC50: >3.75E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128048(US8796328, 26)
Affinity DataIC50: >3.75E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM128035(US8796328, 12)
Affinity DataIC50: >3.75E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In DepthDetails US Patent