Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 6487
TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131882BDBM131882(US8835444, 5.27)
Affinity DataIC50: 13nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131876BDBM131876(US8835444, 5.1)
Affinity DataIC50: 21nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131881BDBM131881(US8835444, 5.26)
Affinity DataIC50: 22nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131860BDBM131860(US8835444, 1.8)
Affinity DataIC50: 35nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131875BDBM131875(US8835444, 4.6)
Affinity DataIC50: 40nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131883BDBM131883(US8835444, 5.29)
Affinity DataIC50: 49nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131872BDBM131872(US8835444, 4.2)
Affinity DataIC50: 59nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131878BDBM131878(US8835444, 5.11)
Affinity DataIC50: 67nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131871BDBM131871(US8835444, 4.1)
Affinity DataIC50: 82nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 9237BDBM9237(US8835444, 4.8 | US8835444, 4.3)
Affinity DataIC50: 88nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131880BDBM131880(US8835444, 5.21)
Affinity DataIC50: 95nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131877BDBM131877(US8835444, 5.8)
Affinity DataIC50: 126nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131863BDBM131863(US8835444, 2.4)
Affinity DataIC50: 131nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131879BDBM131879(US8835444, 5.17)
Affinity DataIC50: 132nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131858BDBM131858(US8835444, 1.1)
Affinity DataIC50: 134nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131869BDBM131869(US8835444, 3.6)
Affinity DataIC50: 142nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131867BDBM131867(US8835444, 2.16)
Affinity DataIC50: 147nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131861BDBM131861(US8835444, 2.0)
Affinity DataIC50: 160nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131864BDBM131864(US8835444, 2.13)
Affinity DataIC50: 167nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131866BDBM131866(US8835444, 2.15)
Affinity DataIC50: 170nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131868BDBM131868(US8835444, 3.3)
Affinity DataIC50: 180nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131865BDBM131865(US8835444, 2.14)
Affinity DataIC50: 214nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 9227BDBM9227(US8835444, 2.1)
Affinity DataIC50: 256nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 9237BDBM9237(US8835444, 4.8 | US8835444, 4.3)
Affinity DataIC50: 262nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131862BDBM131862(US8835444, 2.3)
Affinity DataIC50: 318nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131870BDBM131870(US8835444, 3.17)
Affinity DataIC50: 634nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131874BDBM131874(US8835444, 4.5)
Affinity DataIC50: 665nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131860BDBM131860(US8835444, 1.8)
Affinity DataIC50: 727nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131859BDBM131859(US8835444, 1.4)
Affinity DataIC50: 948nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131882BDBM131882(US8835444, 5.27)
Affinity DataIC50: 2.03E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131869BDBM131869(US8835444, 3.6)
Affinity DataIC50: 3.74E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131868BDBM131868(US8835444, 3.3)
Affinity DataIC50: 4.63E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131880BDBM131880(US8835444, 5.21)
Affinity DataIC50: 4.85E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131858BDBM131858(US8835444, 1.1)
Affinity DataIC50: 4.88E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 2(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131863BDBM131863(US8835444, 2.4)
Affinity DataIC50: 4.94E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent

TargetCorticotropin-releasing factor receptor 1(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 131873BDBM131873(US8835444, 4.4)
Affinity DataIC50: 6.96E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2015
Entry Details
US Patent