Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 6504
TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134267BDBM134267(US8846660, 41)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134262BDBM134262(US8846660, 30)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134278BDBM134278(US8846660, 96)
Affinity DataIC50: 7nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134276BDBM134276(US8846660, 76)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134263BDBM134263(US8846660, 31)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134266BDBM134266(US8846660, 40)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134261BDBM134261(US8846660, 29)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134260BDBM134260(US8846660, 27)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134272BDBM134272(US8846660, 58)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134256BDBM134256(US8846660, 18)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134268BDBM134268(US8846660, 42)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134269BDBM134269(US8846660, 44)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134253BDBM134253(US8846660, 103 | US8846660, 12)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134264BDBM134264(US8846660, 34)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134280BDBM134280(US8846660, 108)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134275BDBM134275(US8846660, 73)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134255BDBM134255(US8846660, 15)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134273BDBM134273(US8846660, 64)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134257BDBM134257(US8846660, 20)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134252BDBM134252(US8846660, 3)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134270BDBM134270(US8846660, 49)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134254BDBM134254(US8846660, 14)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134281BDBM134281(US8846660, 113)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134271BDBM134271(US8846660, 53)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134258BDBM134258(US8846660, 22)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134265BDBM134265(US8846660, 37)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134259BDBM134259(US8846660, 26)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134274BDBM134274(US8846660, 67)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent

TargetChymase(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 134277BDBM134277(US8846660, 88)
Affinity DataIC50: 60nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of the compounds of the present invention for recombinant human chymase was measured by the method of Pasztor et al. (Pasztor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2015
Entry Details
US Patent