Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 6577
LigandChemical structure of BindingDB Monomer ID 139736BDBM139736(US8895549, 11)
Affinity DataIC50: 1.60nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139746BDBM139746(US8895549, 24)
Affinity DataIC50: 1.99nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139750BDBM139750(US8895549, 9)
Affinity DataIC50: 2.02nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139741BDBM139741(US8895549, 7)
Affinity DataIC50: 2.22nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139743BDBM139743(US8895549, 8)
Affinity DataIC50: 2.62nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139754BDBM139754(US8895549, 19)
Affinity DataIC50: 2.78nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139717BDBM139717(US8895549, 2 | US9675616, 2 N-(8-{[(2R)-2-hydroxy-...)
Affinity DataIC50: 2.98nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139763BDBM139763(US8895549, 37)
Affinity DataIC50: 2.98nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139752BDBM139752(US8895549, 14)
Affinity DataIC50: 3.09nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139749BDBM139749(US8895549, 40)
Affinity DataIC50: 3.09nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139747BDBM139747(US8895549, 36)
Affinity DataIC50: 3.41nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139727BDBM139727(US8895549, 5)
Affinity DataIC50: 3.68nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139745BDBM139745(US8895549, 18)
Affinity DataIC50: 3.90nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139729BDBM139729(US8895549, 16)
Affinity DataIC50: 3.94nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139738BDBM139738(US8895549, 20)
Affinity DataIC50: 4.20nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139731BDBM139731(US8895549, 28)
Affinity DataIC50: 4.71nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139737BDBM139737(US8895549, 12)
Affinity DataIC50: 4.74nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139724BDBM139724(US8895549, 4 | US9675616, 4 N-[8-({(2R)-3-[(2R,6S)...)
Affinity DataIC50: 4.85nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139764BDBM139764(US8895549, 39)
Affinity DataIC50: 5.32nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139730BDBM139730(US8895549, 17)
Affinity DataIC50: 5.36nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139735BDBM139735(US8895549, 10)
Affinity DataIC50: 5.47nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139720BDBM139720(US8895549, 27)
Affinity DataIC50: 5.52nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139748BDBM139748(US8895549, 38)
Affinity DataIC50: 5.64nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139740BDBM139740(US8895549, 41)
Affinity DataIC50: 5.83nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139761BDBM139761(US8895549, 32)
Affinity DataIC50: 5.91nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139721BDBM139721(US8895549, 3 | US9675616, 3 N-(8-{[(2S)-2-hydroxy-...)
Affinity DataIC50: 6.20nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139733BDBM139733(US8895549, 35)
Affinity DataIC50: 6.30nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139739BDBM139739(US8895549, 29)
Affinity DataIC50: 6.75nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139732BDBM139732(US8895549, 34)
Affinity DataIC50: 7.21nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139756BDBM139756(US8895549, 23)
Affinity DataIC50: 7.30nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139757BDBM139757(US8895549, 25)
Affinity DataIC50: 8.30nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139759BDBM139759(US8895549, 30)
Affinity DataIC50: 8.83nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139716BDBM139716(US8895549, 21)
Affinity DataIC50: 9.37nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139715BDBM139715(US8895549, Comparative Example 1 | US9675616, 1 N-...)
Affinity DataIC50: 9.92nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 139734BDBM139734(US8895549, 6)
Affinity DataIC50: 9.96nMAssay Description:As reagents for the kinase reaction itself and the quantification of the reaction product, the PI3-Kinase HTRF Assay kit from Millipore (#33-017) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent