Compile Data Set for Download or QSAR
Report error Found 124 Enz. Inhib. hit(s) with all data for entry = 6889
LigandPNGBDBM50398017(CHEMBL2180411 | US9018217, 5,8-Dimethyl-2-[2-(1-me...)
Affinity DataIC50: 0.320nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47287(US9018217, 5,7-Dimethyl-2-[2-(4-phenyl-1-propyl-1H...)
Affinity DataIC50: 0.690nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156359(US9018217, 8-Ethyl-5-methyl-2-[2-(1-methyl-4-pheny...)
Affinity DataIC50: 0.930nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47296(US9018217, 8-Ethyl-5-methyl-2-(2-(1-methyl-4-pheny...)
Affinity DataIC50: 1.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47283(US9018217, 5-Methyl-2-(2-[4-phenyl-1-(2-piperidin-...)
Affinity DataIC50: 1.30nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156347(US9018217, 2-[2-(1-Isobutyl-4-phenyl-1H-imidazol-2...)
Affinity DataIC50: 1.30nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156350(US9018217, 5,7-Dimethyl-2-{2-[1-(2-morpholin-4-yl-...)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156337(US9018217, 2-[2-(1-Isobutyl-4-phenyl-1H-imidazol-2...)
Affinity DataIC50: 1.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM50398014(CHEMBL2180414 | US9018217, 5,8-Dimethyl-2-[2-(1-me...)
Affinity DataIC50: 1.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156352(US9018217, 8-methoxy-5-methyl-2-(2-(1-methyl-4-phe...)
Affinity DataIC50: 2.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156346(US9018217, 5,7-Dimethyl-2-{2-[4-phenyl-1-(2-piperi...)
Affinity DataIC50: 2.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47278(US9018217, 1-Methyl-3-(2-[2-[2-(5-methyl-[1,2,4]tr...)
Affinity DataIC50: 2.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156333(US9018217, 5-Methyl-2-[2-(4-phenyl-1H-imidazol-2-y...)
Affinity DataIC50: 2.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156342(US9018217, 5-Methyl-2-[2-(1-methyl-4-phenyl-1H-imi...)
Affinity DataIC50: 2.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156348(US9018217, 2-[2-(1-Isopropyl-4-phenyl-1H-imidazol-...)
Affinity DataIC50: 3.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156354(US9018217, 5-Methyl-2-[2-(1-methyl-4-phenyl-1H-imi...)
Affinity DataIC50: 3.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156334(US9018217, 2-(1-Isobutyl-4-phenyl-1H-imidazol-2-yl...)
Affinity DataIC50: 4.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47285(US9018217, 1-(2-[2-[2-(5,7-Dimethyl-[1,2,4]triazol...)
Affinity DataIC50: 4.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156356(US9018217, 7-Isopropyl-5-methyl-2-[2-(1-methyl-4-p...)
Affinity DataIC50: 4.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156335(US9018217, 5,7-Dimethyl-2-[1-(2-morpholin-4-yl-eth...)
Affinity DataIC50: 5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156330(US9018217, 5,7-Dimethyl-2-[2-(4-phenyl-1H-imidazol...)
Affinity DataIC50: 5.30nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156255(US9018217, 5,7-Dimethyl-2-[1-(3-methyl-butyl)-4-ph...)
Affinity DataIC50: 5.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156351(US9018217, (S)-1-{2-[2-(5,7-Dimethyl-[1,2,4]triazo...)
Affinity DataIC50: 5.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156324(US9018217, 4-(2-(2-(2-(5,7-dimethyl-[1,2,4]triazol...)
Affinity DataIC50: 6nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156336(US9018217, 5-Methyl-2-[2-(1-methyl-4-phenyl-1H-imi...)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM50398016(CHEMBL2180412 | US9018217, 5,8-Dimethyl-2-[2-(1-me...)
Affinity DataIC50: 7.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47282(US9018217, Diisopropyl-(2-[2-[2-(5-methyl-[1,2,4]t...)
Affinity DataIC50: 7.30nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156344(US9018217, 5-Ethyl-2-(1-methyl-4-phenyl-1H-imidazo...)
Affinity DataIC50: 7.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47276(US9018217, 1-Methyl-3-(2-[2-[2-(5-methyl-[1,2,4]tr...)
Affinity DataIC50: 8.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156322(US9018217, 5-Methyl-2-{2-[1-(2-morpholin-4-yl-ethy...)
Affinity DataIC50: 8.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156349(US9018217, (2-{2-[2-(5,7-Dimethyl-[1,2,4]triazolo[...)
Affinity DataIC50: 8.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156256(US9018217, 5,7-Dimethyl-2-(4-phenyl-1-propyl-1H-im...)
Affinity DataIC50: 9.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47289(US9018217, (R)-1-[2-[2-(5,7-Dimethyl-[1,2,4]triazo...)
Affinity DataIC50: 11nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156257(US9018217, 2-(1-Cyclopropylmethyl-4-phenyl-1H-imid...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156320(US9018217, 8-Methyl-2-[2-(1-methyl-4-phenyl-1H-Imi...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156327(US9018217, 5,7-Dimethyl-2-[2-(1-methyl-4-phenyl-1H...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47288(US9018217, 1-[2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1...)
Affinity DataIC50: 13nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156321(US9018217, 5-Methyl-2-[2-(1-methyl-4-phenyl-1H-imi...)
Affinity DataIC50: 14nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156326(US9018217, 5,7-dimethyl-2-(2-(4-phenyl-1H-imidazol...)
Affinity DataIC50: 15nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156341(US9018217, 5,6,7-Trimethyl-2-[2-(1-methyl-4-phenyl...)
Affinity DataIC50: 15nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156358(US9018217, {5-Methyl-2-[2-(1-methyl-4-phenyl-1H-im...)
Affinity DataIC50: 15nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47274(US9018217, 4-(2-(2-((8-chloro-[1,2,4]triazolo[1,5-...)
Affinity DataIC50: 17nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM50398015(CHEMBL2180413 | US9018217, 5,7-dimethyl-2-(2-(1-me...)
Affinity DataIC50: 17nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156325(US9018217, 6,8-dimethyl-2-(2-(1-methyl-4-phenyl-1H...)
Affinity DataIC50: 19nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156258(US9018217, 5,7-dimethyl-2((1-methyl-4-phenyl-1H-im...)
Affinity DataIC50: 20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156259(US9018217, 5,7-Dimethyl-2-[1-(2-morpholin-4-yl-eth...)
Affinity DataIC50: 22nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156338(US9018217, 2-[2-(1-Isopropyl-4-phenyl-1H-imidazol-...)
Affinity DataIC50: 23nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156331(US9018217, 5,7-Dimethyl-2-(4-phenyl-1H-imidazol-2-...)
Affinity DataIC50: 24nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM47281(US9018217, 5-Methyl-2-{2-[4-phenyl-1-(3-piperidin-...)
Affinity DataIC50: 25nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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LigandPNGBDBM156332(US9018217, 5,7-Dimethyl-2-(1-methyl-4-phenyl-1H-im...)
Affinity DataIC50: 25nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
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