Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 6932
TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160321BDBM160321(US9040693, 22)
Affinity DataIC50: 2nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160326BDBM160326(US9040693, 146)
Affinity DataIC50: 10nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160329BDBM160329(US9040693, 233)
Affinity DataIC50: 15nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160330BDBM160330(US9040693, 367)
Affinity DataIC50: 15nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160327BDBM160327(US9040693, 191)
Affinity DataIC50: 17nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160325BDBM160325(US9040693, 95)
Affinity DataIC50: 19nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160328BDBM160328(US9040693, 202)
Affinity DataIC50: 20nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160332BDBM160332(US9040693, 420)
Affinity DataIC50: 29nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160324BDBM160324(US9040693, 48)
Affinity DataIC50: 29nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160331BDBM160331(US9040693, 414)
Affinity DataIC50: 42nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160319BDBM160319(US9040693, 3)
Affinity DataIC50: 80nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160322BDBM160322(US9040693, 25)
Affinity DataIC50: 85nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160320BDBM160320(US9040693, 17)
Affinity DataIC50: 101nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160318BDBM160318(US9040693, 2)
Affinity DataIC50: 199nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 160323BDBM160323(US9040693, 31)
Affinity DataIC50: 272nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent