Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 6968
Affinity DataKi: 33.1nM ΔG°: -42.7kJ/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair
Affinity DataKi: 42.5nM ΔG°: -42.1kJ/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair
Affinity DataKi: 64.5nM ΔG°: -41.0kJ/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair
Affinity DataKi: 66.8nM ΔG°: -41.0kJ/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair
Affinity DataKi: 79.1nM ΔG°: -40.5kJ/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair
Affinity DataKi: 89.6nM ΔG°: -40.2kJ/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair
Affinity DataKi: 621nM ΔG°: -38.4kJ/molepH: 7.4 T: 50°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataKi: 853nM ΔG°: -37.5kJ/molepH: 7.4 T: 50°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataKi: 977nM ΔG°: -37.2kJ/molepH: 7.4 T: 50°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataKi: 1.34E+3nM ΔG°: -36.3kJ/molepH: 7.4 T: 50°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataIC50: 66.8nMpH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant ...More data for this Ligand-Target Pair