Compile Data Set for Download or QSAR
maximum 50k data
Found 130 Enz. Inhib. hit(s) with all data for entry = 7066
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172187(US9090564, 1)
Affinity DataIC50:  0.660nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172221(US9090564, 35)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172197(US9090564, 11 | US9096594, 54)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172194(US9090564, 8)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172262(US9090564, 76)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172267(US9090564, 81)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172266(US9090564, 80)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172265(US9090564, 79)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172260(US9090564, 74)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172259(US9090564, 73)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172268(US9090564, 82)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172269(US9090564, 83)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172224(US9090564, 38)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172216(US9090564, 30)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172212(US9090564, 26)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172188(US9090564, 2)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172196(US9090564, 10 | US9096594, 22)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172225(US9090564, 39)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172297(US9090564, 111)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172200(US9090564, 14)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172264(US9090564, 78)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172247(US9090564, 61)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172316(US9090564, 130)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172210(US9090564, 24)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172246(US9090564, 60)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172277(US9090564, 91)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172193(US9090564, 7)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172290(US9090564, 104)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172276(US9090564, 90)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172228(US9090564, 42)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172298(US9090564, 112)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172220(US9090564, 34)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172274(US9090564, 88)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172195(US9090564, 9)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172211(US9090564, 25)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172234(US9090564, 48)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172239(US9090564, 53)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172223(US9090564, 37)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172204(US9090564, 18)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172192(US9090564, 6)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172232(US9090564, 46)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172300(US9090564, 114)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172299(US9090564, 113)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172286(US9090564, 100)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172273(US9090564, 87)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172271(US9090564, 85)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172215(US9090564, 29)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172236(US9090564, 50)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172231(US9090564, 45)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM172282(US9090564, 96)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Kinase reaction conditions:400 nM GFP-4E-BP1, 8 uM ATP, -150 ng/mL mTOR, 50 mM HEPES pH 7.5, 0.01% Polysorbate 20, 1 mM EGTA, 10 mM MnC12, and variab...More data for this Ligand-Target Pair
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