Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 7079
LigandPNGBDBM173175(US9096589, 8-Methoxy-5-methyl-2-{2-[1-(2-morpholin...)
Affinity DataIC50: 0.330nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173179(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiophen-...)
Affinity DataIC50: 0.390nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173191(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiazol-4...)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173192(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-pyrimidin...)
Affinity DataIC50: 0.440nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173193(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-pyrazin-2...)
Affinity DataIC50: 0.520nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173112(US9096589, 5-Methyl-2-[2-(4-thiophen-2-yl-1H-imida...)
Affinity DataIC50: 0.540nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173194(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-pyridin-4...)
Affinity DataIC50: 0.550nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173113(US9096589, 8-Methyl-2-[2-(4-thiophen-2-yl-1H-imida...)
Affinity DataIC50: 0.990nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173171(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiophen-...)
Affinity DataIC50: 1nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173170(US9096589, 8-Methoxy-5-methyl-2-[2-(4-thiophen-2-y...)
Affinity DataIC50: 1.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173172(US9096589, 8-Methoxy-5-methyl-2-[2-(1-propyl-4-thi...)
Affinity DataIC50: 1.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173190(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiazol-4...)
Affinity DataIC50: 1.29nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173140(US9096589, 8-Methoxy-5-methyl-2-[2-(1-methyl-4-thi...)
Affinity DataIC50: 1.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173176(US9096589, 8-Methoxy-5-methyl-2-[2-(1-methyl-4-thi...)
Affinity DataIC50: 1.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173174(US9096589, 4-{2-[2-(8-Methoxy-5-methyl-[1,2,4]tria...)
Affinity DataIC50: 1.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173180(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiazol-2...)
Affinity DataIC50: 2.30nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173129(US9096589, 8-Methoxy-5-methyl-2-[(E)-2-(1-methyl-4...)
Affinity DataIC50: 2.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173181(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiazol-2...)
Affinity DataIC50: 2.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173137(US9096589, (R)-1-Chloro-3-{2-[2-(5-methyl-[1,2,4]t...)
Affinity DataIC50: 2.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173187(US9096589, 2-[2-(4-Furan-3-yl-1-methyl-1H-imidazol...)
Affinity DataIC50: 2.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173182(US9096589, 8-Methoxy-5-methyl-2-{2-[1-methyl-4-(4-...)
Affinity DataIC50: 3.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173102(US9669029, 23 5,7-Dimethyl-2-[2-(1-propyl-4-thioph...)
Affinity DataIC50: 3.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173177(US9096589, 2-[2-(4-Furan-3-yl-1-methyl-1H-imidazol...)
Affinity DataIC50: 4nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173173(US9096589, 8-Methoxy-5-methyl-2-[2-(1-prop-2-ynyl-...)
Affinity DataIC50: 4.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173130(US9096589, 5,7-Dimethyl-2-[2-(1-methyl-4-thiophen-...)
Affinity DataIC50: 4.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173185(US9096589, 5,8-Dimethyl-2-{2-[1-methyl-4-(5-methyl...)
Affinity DataIC50: 4.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173131(US9096589, 8-Methoxy-2-[2-(1-methyl-4-thiophen-2-y...)
Affinity DataIC50: 4.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173111(US9096589, 1-(4-Chloro-phenyl)-2-{2-[2-(5,7-dimeth...)
Affinity DataIC50: 5.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173119(US9096589, 5-Methyl-2-[2-(4-thiophen-3-yl-1H-imida...)
Affinity DataIC50: 5.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173183(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-pyridin-3...)
Affinity DataIC50: 5.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173114(US9096589, (S)-2-{2-[2-(5-Methyl-[1,2,4]triazolo[1...)
Affinity DataIC50: 6.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173178(US9096589, 5,8-Dimethyl-2-{2-[1-methyl-4-(5-methyl...)
Affinity DataIC50: 6.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173105(US9669029, 26 5,7-Dimethyl-2-{2-[1-(3-methyl-butyl...)
Affinity DataIC50: 6.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173189(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiazol-5...)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173115(US9096589, 1-Methoxy-3-{2-[2-(5-methyl-[1,2,4]tria...)
Affinity DataIC50: 7.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173096(US9669029, 17 5,7-Dimethyl-2-[2-(4-thiophen-2-yl-1...)
Affinity DataIC50: 7.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173101(US9096589, 1-{2-[2-(5,7-Dimethyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 7.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173161(US9096589, 1-Methoxy-3-{2-[2-(8-methyl-[1,2,4]tria...)
Affinity DataIC50: 8.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173153(US9096589, [((S)-2-Hydroxy-3-{2-[2-(5-methyl-[1,2,...)
Affinity DataIC50: 8.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173100(US9669029, 21 (S)-2-{2-[2-(5,7-Dimethyl-imidazo[1,...)
Affinity DataIC50: 8.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173083(US9669029, 3 5,7-Dimethyl-2-[(E)-2-(1-methyl-4-thi...)
Affinity DataIC50: 8.80nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173184(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-pyridin-3...)
Affinity DataIC50: 8.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173162(US9096589, 5-Methyl-2-[2-(1-methyl-4-thiophen-2-yl...)
Affinity DataIC50: 9.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173168(US9096589, 8-Methoxy-5-methyl-2-[2-(1-methyl-4-thi...)
Affinity DataIC50: 9.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173095(US9096589, 5,7-Dimethyl-2-{2-[4-thiophen-2-yl-1-(2...)
Affinity DataIC50: 9.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173120(US9096589, 5-Methyl-2-[2-(4-pyridin-3-yl-1H-imidaz...)
Affinity DataIC50: 9.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173120(US9096589, 5-Methyl-2-[2-(4-pyridin-3-yl-1H-imidaz...)
Affinity DataIC50: 9.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM60522(US9096589, 5,8-Dimethyl-2-[2-(1-methyl-4-thiazol-2...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173106(US9096589, 2-[2-(1-Isobutyl-4-thiophen-2-yl-1H-imi...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

LigandPNGBDBM173108(US9669029, 29 1-{2-[2-(5,7-Dimethyl-imidazo[1,2-a]...)
Affinity DataIC50: 14nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent

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