Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 7105
TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174845(US9115061, XII)
Affinity DataKd:  40nMpH: 7.4Assay Description:Titrations were performed using a VP-ITC or ITC200 calorimeter from Microcal (Northampton, Mass.). BCL-XL was used at concentrations between 25 and 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174848(US9115061, XVI)
Affinity DataIC50: 140nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174843(US9115061, VIII)
Affinity DataIC50: 160nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174838(US9115061, I)
Affinity DataKd:  170nMpH: 7.4Assay Description:Titrations were performed using a VP-ITC or ITC200 calorimeter from Microcal (Northampton, Mass.). BCL-XL was used at concentrations between 25 and 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174838(US9115061, I)
Affinity DataIC50: 190nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174844(US9115061, XI)
Affinity DataIC50: 250nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174845(US9115061, XII)
Affinity DataIC50: 320nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174841(US9115061, VI)
Affinity DataIC50: 450nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174840(US9115061, V)
Affinity DataIC50: 1.29E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174839(US9115061, IV)
Affinity DataIC50: 1.30E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174847(US9115061, XIV)
Affinity DataIC50: 1.30E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174846(US9115061, XIII)
Affinity DataIC50: 1.31E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM31802(Apogossypol | US9115061, Apogossypol)
Affinity DataKd:  1.70E+3nMpH: 7.4Assay Description:Titrations were performed using a VP-ITC or ITC200 calorimeter from Microcal (Northampton, Mass.). BCL-XL was used at concentrations between 25 and 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 2.72E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174843(US9115061, VIII)
Affinity DataKd:  2.75E+3nMpH: 7.4Assay Description:Titrations were performed using a VP-ITC or ITC200 calorimeter from Microcal (Northampton, Mass.). BCL-XL was used at concentrations between 25 and 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174842(US9115061, VII)
Affinity DataIC50: 2.90E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent

TargetBcl-2-like protein 1(Human)
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM31802(Apogossypol | US9115061, Apogossypol)
Affinity DataIC50: 3.69E+3nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details
US Patent