Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 7139
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177755(US9120781, 18)
Affinity DataKi:  0.130nM ΔG°:  -56.4kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177758(US9120781, 26)
Affinity DataKi:  0.200nM ΔG°:  -55.4kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177756(US9120781, 22)
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177753(US9120781, 9)
Affinity DataKi:  0.600nM ΔG°:  -52.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177759(US9120781, 32)
Affinity DataKi:  2.5nM ΔG°:  -49.1kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177754(US9120781, 13)
Affinity DataKi:  7.40nM ΔG°:  -46.4kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

US Patent
LigandPNGBDBM177757(US9120781, 23)
Affinity DataKi:  484nM ΔG°:  -36.0kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent