Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 7200
TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180890BDBM180890(US9133182, Example 19)
Affinity DataIC50: 4nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180896BDBM180896(US9133182, Example 25)
Affinity DataIC50: 10nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180874BDBM180874(US9133182, Example 3)
Affinity DataIC50: 11nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180884BDBM180884(US9133182, Example 13)
Affinity DataIC50: 13nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180888BDBM180888(US9133182, Example 17)
Affinity DataIC50: 13nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180872BDBM180872(US9133182, Example 1)
Affinity DataIC50: 14nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180892BDBM180892(US9133182, Example 21)
Affinity DataIC50: 15nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180900BDBM180900(US9133182, Example 29)
Affinity DataIC50: 25nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180882BDBM180882(US9133182, Example 11)
Affinity DataIC50: 25nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180894BDBM180894(US9133182, Example 23)
Affinity DataIC50: 33nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180880BDBM180880(US9133182, Example 9)
Affinity DataIC50: 45nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180902BDBM180902(US9133182, Example 31)
Affinity DataIC50: 46nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180878BDBM180878(US9133182, Example 7)
Affinity DataIC50: 50nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180898BDBM180898(US9133182, Example 27)
Affinity DataIC50: 62nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180903BDBM180903(US9133182, Example 33)
Affinity DataIC50: 65nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180891BDBM180891(US9133182, Example 20)
Affinity DataIC50: 72nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180873BDBM180873(US9133182, Example 2)
Affinity DataIC50: 100nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180875BDBM180875(US9133182, Example 4)
Affinity DataIC50: 120nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180908BDBM180908(US9133182, Example 38)
Affinity DataIC50: 150nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180886BDBM180886(US9133182, Example 15)
Affinity DataIC50: 200nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180893BDBM180893(US9133182, Example 22)
Affinity DataIC50: 210nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180901BDBM180901(US9133182, Example 30)
Affinity DataIC50: 491nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180876BDBM180876(US9133182, Example 5)
Affinity DataIC50: 530nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180909BDBM180909(US9133182, Example 39)
Affinity DataIC50: 550nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180889BDBM180889(US9133182, Example 18)
Affinity DataIC50: 700nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180883BDBM180883(US9133182, Example 12)
Affinity DataIC50: 933nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180899BDBM180899(US9133182, Example 28)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180885BDBM180885(US9133182, Example 14)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180879BDBM180879(US9133182, Example 8)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180895BDBM180895(US9133182, Example 24)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180881BDBM180881(US9133182, Example 10)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180897BDBM180897(US9133182, Example 26)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180907BDBM180907(US9133182, Example 37)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180904BDBM180904(US9133182, Example 34)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180887BDBM180887(US9133182, Example 16)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180906BDBM180906(US9133182, Example 36)
Affinity DataIC50: 1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAndrogen receptor(Rat)
Radius Health

US Patent
LigandChemical structure of BindingDB Monomer ID 180905BDBM180905(US9133182, Example 35)
Affinity DataIC50: 1.00E+4nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent