Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 7251
TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184568(US9150583, 5)
Affinity DataIC50: 9nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184570(US9150583, 7)
Affinity DataIC50: 11nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184566(US9150583, 3)
Affinity DataIC50: 11nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184564(US9150583, 1)
Affinity DataIC50: 15nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184565(US9150583, 2)
Affinity DataIC50: 18nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184569(US9150583, 6)
Affinity DataIC50: 43nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184567(US9150583, 4)
Affinity DataIC50: 90nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent

TargetCholesteryl ester transfer protein(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184571(US9150583, 8)
Affinity DataIC50: 210nMT: 2°CAssay Description:CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
US Patent